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Cardioselective beta blockers

What are Cardioselective beta blockers?

Beta-adrenergic blocking agents prevent stimulation of the beta-1 adrenergic receptors at the nerve endings of the sympathetic nervous system and therefore decrease the activity of the heart. They block sympathetic stimulation of the heart and reduce systolic pressure, heart rate, cardiac contractility and output, which in turn decreases the demand by the heart for oxygen and increases exercise tolerance. Beta-adrenergic blocking agents may also affect beta-2 adrenergic receptors located in the bronchial smooth muscle of the airways, which has the potential to cause bronchoconstriction (a narrowing of the breathing passages).

Cardioselective beta blockers have a clinical advantage in that they are 20 times more potent at blocking beta-1 receptors than beta-2 receptors. They are therefore less likely to cause bronchoconstriction compared with non-selective beta-blockers; however, the danger of bronchoconstriction cannot be totally ignored, as they are not totally selective.

Beta-adrenergic blocking agents are used to treat angina, control abnormal heart rhythms and to reduce high blood pressure.

List of Cardioselective beta blockers:

View by  Brand | Generic
Drug Name Reviews Avg. Ratings
Kerlone (Pro)
Generic name: betaxolol
0 reviews
Sectral (Pro)
Generic name: acebutolol
3 reviews
Brevibloc (Pro)
Generic name: esmolol
0 reviews
Tenormin (Pro)
Generic name: atenolol
26 reviews
Zebeta (Pro)
Generic name: bisoprolol
3 reviews
Toprol-XL (Pro)
Generic name: metoprolol
52 reviews
Lopressor (Pro)
Generic name: metoprolol
13 reviews
Bystolic (Pro)
Generic name: nebivolol
200 reviews
For ratings, users were asked how effective they found the medicine while considering positive/adverse effects and ease of use (1 = not effective, 10 = most effective).

Further information

Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.