Narcotic analgesics

A drug may be classified by the chemical type of the active ingredient or by the way it is used to treat a particular condition. Each drug can be classified into one or more drug classes.

Narcotic analgesics are drugs that relieve pain, can cause numbness and induce a state of unconsciousness.

They work by binding to opioid receptors, which are present in the central and peripheral nervous system. There are three types of opioid receptors, which are all G-protein linked and either facilitate opening of potassium channels (causing hyperpolarization) or inhibit calcium channel opening (so inhibits release of excitatory neurotransmitters such as substance P). Overall, narcotic analgesics reduce neuronal excitability in the pain carrying pathway.

Morphine and its analogues, and some synthetic derivatives are classed as narcotics analgesics. Narcotic analgesics are used to relieve acute and chronic, severe pain. Some narcotics are more potent than others. They also have the tendency to cause tolerance and dependence.

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Drug Name DownUp( View by: Brand | Generic ) Reviews Avg. Ratings DownUp
Alfenta (More...)
generic name: alfentanil
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10
Astramorph PF (Pro, More...)
generic name: morphine
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10
Ionsys (Pro, More...)
generic name: fentanyl
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10
Levo-Dromoran (Pro, More...)
generic name: levorphanol
2 Review(s)
  
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10
Numorphan (Pro, More...)
generic name: oxymorphone
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10
Onsolis (Pro, More...)
generic name: fentanyl
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10
Oxyfast (More...)
generic name: oxycodone
1 Review(s)
  
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10
Roxanol (More...)
generic name: morphine
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10
Roxanol-T (More...)
generic name: morphine
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10
Roxicodone Intensol (More...)
generic name: oxycodone
3 Review(s)
  
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10
Meperitab (More...)
generic name: meperidine
3 Review(s)
  
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9.8
Sublimaze (Pro, More...)
generic name: fentanyl
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9.8
Actiq (Pro, More...)
generic name: fentanyl
10 Review(s)
  
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9.4
Methadone Diskets (More...)
generic name: methadone
10 Review(s)
  
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9.4
Subutex (More...)
generic name: buprenorphine
38 Review(s)
  
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9.4
Duragesic-50 (More...)
generic name: fentanyl
3 Review(s)
  
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9.3
Fentora (Pro, More...)
generic name: fentanyl
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9.3
Duragesic-25 (More...)
generic name: fentanyl
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9.2
Abstral (Pro, More...)
generic name: fentanyl
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9.0
Demerol (Pro, More...)
generic name: meperidine
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9.0
Dolophine (Pro, More...)
generic name: methadone
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9.0
Nucynta ER (Pro, More...)
generic name: tapentadol
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9.0
Oxydose (More...)
generic name: oxycodone
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9.0
Roxicodone (Pro, More...)
generic name: oxycodone
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9.0
Methadose (Pro, More...)
generic name: methadone
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8.9
Dilaudid (Pro, More...)
generic name: hydromorphone
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8.8
MSIR (More...)
generic name: morphine
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8.8
OxyContin (Pro, More...)
generic name: oxycodone
168 Review(s)
  
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8.8
Stadol (Pro, More...)
generic name: butorphanol
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8.7
Opana ER (Pro, More...)
generic name: oxymorphone
43 Review(s)
  
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8.5
Duragesic-100 (More...)
generic name: fentanyl
5 Review(s)
  
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8.4
Kadian (Pro, More...)
generic name: morphine
30 Review(s)
  
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8.4
MS Contin (Pro, More...)
generic name: morphine
35 Review(s)
  
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8.4
Opana (Pro, More...)
generic name: oxymorphone
56 Review(s)
  
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8.4
Talwin (More...)
generic name: pentazocine
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8.4
Duragesic (Pro, More...)
generic name: fentanyl
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8.3
Dilaudid-HP (Pro, More...)
generic name: hydromorphone
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8.2
Fentanyl Transdermal System (More...)
generic name: fentanyl
19 Review(s)
  
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8.1
Paregoric (More...)
generic name: opium
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8.1
Duragesic-75 (More...)
generic name: fentanyl
7 Review(s)
  
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8.0
Opium Deodorized (More...)
generic name: opium
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8.0
Avinza (Pro, More...)
generic name: morphine
28 Review(s)
  
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7.9
OxyIR (More...)
generic name: oxycodone
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7.8
Butrans (Pro, More...)
generic name: buprenorphine
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7.7
Nubain (Pro, More...)
generic name: nalbuphine
15 Review(s)
  
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7.7
Buprenex (Pro, More...)
generic name: buprenorphine
2 Review(s)
  
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7.5
Duramorph (Pro, More...)
generic name: morphine
3 Review(s)
  
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7.0
Nucynta (Pro, More...)
generic name: tapentadol
92 Review(s)
  
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7.0
Darvon (Pro, More...)
generic name: propoxyphene
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6.0
Darvon-N (Pro, More...)
generic name: propoxyphene
1 Review(s)
  
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6.0
Oramorph SR (Pro, More...)
generic name: morphine
3 Review(s)
  
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5.8
Duragesic-12 (More...)
generic name: fentanyl
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5.0
Exalgo (Pro, More...)
generic name: hydromorphone
4 Review(s)
  
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5.0
Dazidox (More...)
generic name: oxycodone
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0.0
DepoDur (More...)
generic name: morphine liposomal
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0.0
ETH-Oxydose (More...)
generic name: oxycodone
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0.0
Infumorph (More...)
generic name: morphine
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0.0
Lazanda (More...)
generic name: fentanyl
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0.0
Orlaam (More...)
generic name: levomethadyl acetate
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0.0
Oxecta (Pro, More...)
generic name: oxycodone
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0.0
Palladone (Pro, More...)
generic name: hydromorphone
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0.0
Percolone (More...)
generic name: oxycodone
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0.0
PP-Cap (More...)
generic name: propoxyphene
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0.0
RMS (More...)
generic name: morphine
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0.0
Subsys (More...)
generic name: fentanyl
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0.0
Sufenta (Pro, More...)
generic name: sufentanil
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0.0
Ultiva (Pro, More...)
generic name: remifentanil
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0.0

See also

Medical conditions associated with narcotic analgesics:

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