Alpelisib Drug Interactions
Currently displaying a list of 338 drugs known to interact with alpelisib.
- 15 major drug interactions
- 319 moderate drug interactions
- 4 minor drug interactions
Medications known to interact with alpelisib
Note: Showing generic names only.
A
- abametapir topical
- abrocitinib
- acalabrutinib
- acarbose
- acetohexamide
- adagrasib
- afatinib
- albiglutide
- alendronate
- aliskiren
- alogliptin
- alosetron
- aminoglutethimide
- amitriptyline
- amobarbital
- apalutamide
- apixaban
- armodafinil
- artesunate
- atezolizumab
- atorvastatin
- avelumab
B
- belinostat
- belzutifan
- berotralstat
- betrixaban
- bexagliflozin
- bexarotene
- bortezomib
- bosentan
- bosutinib
- brentuximab
- brigatinib
- bupropion
- butabarbital
- butalbital
C
- canagliflozin
- candesartan
- capivasertib
- carbamazepine
- carvedilol
- celecoxib
- cemiplimab
- cenobamate
- ceritinib
- chlorpropamide
- cladribine
- cobicistat
- cobimetinib
- colchicine
- cosibelimab
- cyclophosphamide
- cyclosporine
D
- dabigatran
- daclatasvir
- danicopan
- dapagliflozin
- dapsone
- daridorexant
- darolutamide
- daunorubicin
- daunorubicin liposomal
- deferasirox
- delafloxacin
- denosumab
- deucravacitinib
- diazepam
- diclofenac
- digoxin
- diltiazem
- docetaxel
- doravirine
- dostarlimab
- doxepin
- doxorubicin
- doxorubicin liposomal
- dronabinol
- dulaglutide
- durvalumab
E
- edaravone
- edoxaban
- efavirenz
- elacestrant
- elafibranor
- elagolix
- eltrombopag
- empagliflozin
- enasidenib
- encorafenib
- entrectinib
- enzalutamide
- epirubicin
- erlotinib
- ertugliflozin
- eslicarbazepine
- etidronate
- etoposide
- etravirine
- everolimus
- exenatide
F
- felbamate
- fenfluramine
- fexinidazole
- fidaxomicin
- fluoxetine
- flurbiprofen
- fluvastatin
- fosphenytoin
- fostemsavir
- futibatinib
G
- gefitinib
- gilteritinib
- glasdegib
- glimepiride
- glipizide
- glyburide
- glycerol phenylbutyrate
- griseofulvin
H
I
- ibandronate
- ibrutinib
- ibuprofen
- idarubicin
- idelalisib
- ifosfamide
- imatinib
- indacaterol
- indomethacin
- insulin
- insulin aspart
- insulin aspart protamine
- insulin degludec
- insulin detemir
- insulin glargine
- insulin glulisine
- insulin inhalation, rapid acting
- insulin isophane
- insulin lispro
- insulin lispro protamine
- insulin regular
- insulin zinc
- insulin zinc extended
- ipilimumab
- iptacopan
- irbesartan
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isotretinoin
- ivacaftor
- ivosidenib
K
L
- lapatinib
- larotrectinib
- lasmiditan
- lazertinib
- lenalidomide
- leniolisib
- lesinurad
- letermovir
- linagliptin
- liraglutide
- lixisenatide
- lonapegsomatropin
- lorlatinib
- losartan
- lovastatin
- lurasidone
- lusutrombopag
M
- maraviroc
- maribavir
- mavacamten
- mavorixafor
- mefenamic acid
- meloxicam
- meperidine
- mephenytoin
- mephobarbital
- meropenem
- metformin
- methadone
- methotrexate
- metreleptin
- midostaurin
- miglitol
- mitapivat
- mitomycin
- mitotane
- mitoxantrone
- mobocertinib
- momelotinib
- montelukast
- morphine
N
- naldemedine
- naloxegol
- naproxen
- nateglinide
- nevirapine
- nicotine
- nilotinib
- nintedanib
- niraparib
- nivolumab
O
P
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palbociclib
- pamidronate
- pantoprazole
- pazopanib
- pembrolizumab
- pentobarbital
- pexidartinib
- phenobarbital
- phenylbutazone
- phenytoin
- pioglitazone
- pirfenidone
- piroxicam
- pirtobrutinib
- ponatinib
- posaconazole
- pralsetinib
- pramlintide
- pretomanid
- primidone
- propofol
- prucalopride
Q
R
- ramelteon
- ranolazine
- regorafenib
- relugolix
- repaglinide
- repotrectinib
- resmetirom
- retifanlimab
- ribociclib
- rifabutin
- rifampin
- rifapentine
- rifaximin
- rimegepant
- riociguat
- ripretinib
- risedronate
- ritlecitinib
- ritonavir
- rivaroxaban
- rolapitant
- romidepsin
- rosiglitazone
- rosuvastatin
- rucaparib
- rufinamide
S
- safinamide
- saquinavir
- saxagliptin
- secobarbital
- seladelpar
- selegiline
- semaglutide
- sertraline
- sildenafil
- silodosin
- simvastatin
- siponimod
- sirolimus
- sitagliptin
- somapacitan-beco
- somatrem
- somatrogon
- somatropin
- sonidegib
- sotagliflozin
- sotorasib
- sparsentan
- st. john's wort
- sulfamethoxazole
- sulfasalazine
- sulfinpyrazone
- suzetrigine
T
- tacrolimus
- talazoparib
- tamoxifen
- tecovirimat
- tedizolid
- telotristat
- teniposide
- tenofovir alafenamide
- tenofovir disoproxil
- tepotinib
- terbinafine
- teriflunomide
- thiotepa
- tiludronate
- tipranavir
- tirzepatide
- tislelizumab
- tivozanib
- tolazamide
- tolbutamide
- tolvaptan
- topotecan
- toripalimab
- torsemide
- tovorafenib
- tremelimumab
- trofinetide
- troglitazone
U
V
- vadadustat
- valdecoxib
- vardenafil
- vemurafenib
- venetoclax
- verapamil
- vimseltinib
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- vorasidenib
- voriconazole
W
Z
Alpelisib alcohol/food interactions
There are 2 alcohol/food interactions with alpelisib.
Alpelisib disease interactions
There are 6 disease interactions with alpelisib which include:
More about alpelisib
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- Drug class: PI3K inhibitors
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.