Pexidartinib Interactions
There are 644 drugs known to interact with pexidartinib, along with 2 disease interactions, and 2 alcohol/food interactions. Of the total drug interactions, 422 are major, 206 are moderate, and 16 are minor.
- View pexidartinib alcohol/food interactions (2)
- View pexidartinib disease interactions (2)
Medications known to interact with pexidartinib
Note: Showing generic names only.
- abacavir
- abametapir topical
- abemaciclib
- abiraterone
- abrocitinib
- acalabrutinib
- acarbose
- acetaminophen
- acitretin
- adagrasib
- ado-trastuzumab emtansine
- afatinib
- aldesleukin
- alectinib
- alfentanil
- allopurinol
- alpelisib
- aluminum carbonate
- aluminum hydroxide
- ambrisentan
- aminosalicylic acid
- amiodarone
- amprenavir
- apalutamide
- apixaban
- apremilast
- aprepitant
- aprocitentan
- aripiprazole
- armodafinil
- asenapine
- ashwaganda
- asparaginase erwinia chrysanthemi
- asparaginase escherichia coli
- astemizole
- atazanavir
- atezolizumab
- atogepant
- atomoxetine
- atorvastatin
- atovaquone
- atrasentan
- avacopan
- avanafil
- avapritinib
- avatrombopag
- avelumab
- axitinib
- azithromycin
- bedaquiline
- belinostat
- belumosudil
- belzutifan
- benazepril
- berotralstat
- bexarotene
- bicalutamide
- binimetinib
- black cohosh
- blinatumomab
- boceprevir
- bortezomib
- bosentan
- bosutinib
- brentuximab
- brexpiprazole
- brigatinib
- brincidofovir
- bromfenac
- bromocriptine
- budesonide
- buprenorphine
- bupropion
- buspirone
- butorphanol
- cabazitaxel
- cabozantinib
- calaspargase pegol
- calcium carbonate
- cannabidiol
- capivasertib
- capmatinib
- captopril
- carbamazepine
- carfilzomib
- cariprazine
- carmustine
- caspofungin
- celecoxib
- cemiplimab
- cenobamate
- ceritinib
- cerivastatin
- cevimeline
- chaparral
- chenodiol
- chloramphenicol
- chlorotrianisene
- chlorzoxazone
- cimetidine
- cinacalcet
- ciprofloxacin
- cisapride
- clarithromycin
- clavulanate
- clobazam
- clofarabine
- clofazimine
- clopidogrel
- clotrimazole
- cobicistat
- cobimetinib
- comfrey
- conivaptan
- conjugated estrogens
- copanlisib
- cosibelimab
- crinecerfont
- crizotinib
- cyclosporine
- cytarabine
- dabrafenib
- dacarbazine
- daclatasvir
- daclizumab
- dacomitinib
- danazol
- danicopan
- dantrolene
- dapsone topical
- daridorexant
- darifenacin
- darolutamide
- darunavir
- dasatinib
- deferasirox
- deflazacort
- dehydroepiandrosterone
- delandistrogene moxeparvovec
- delavirdine
- deucravacitinib
- dexamethasone
- dexlansoprazole
- diclofenac
- diclofenac topical
- didanosine
- dihydroergotamine
- dihydroxyaluminum sodium carbonate
- diltiazem
- dimethyl fumarate
- diroximel fumarate
- disulfiram
- divalproex sodium
- docetaxel
- dolutegravir
- donepezil
- doravirine
- dostarlimab
- doxazosin
- doxercalciferol
- doxorubicin
- doxorubicin liposomal
- doxycycline
- dronedarone
- droperidol
- drospirenone
- duloxetine
- durvalumab
- duvelisib
- efavirenz
- eflornithine
- elacestrant
- elagolix
- eliglustat
- elotuzumab
- elranatamab
- eltrombopag
- elvitegravir
- emtricitabine
- enalapril
- enalaprilat
- encorafenib
- enfortumab vedotin
- entrectinib
- enzalutamide
- epirubicin
- erdafitinib
- ergonovine
- ergotamine
- erlotinib
- erythromycin
- eslicarbazepine
- esomeprazole
- estazolam
- esterified estrogens
- estradiol
- estrone
- estropipate
- eszopiclone
- ethambutol
- ethanol
- ethinyl estradiol
- ethionamide
- ethotoin
- etodolac
- etonogestrel
- etranacogene dezaparvovec
- etrasimod
- etravirine
- etretinate
- everolimus
- exemestane
- ezetimibe
- famotidine
- febuxostat
- fedratinib
- felbamate
- fenfluramine
- fenofibrate
- fenofibric acid
- fenoprofen
- fentanyl
- fesoterodine
- fexinidazole
- fezolinetant
- fidanacogene elaparvovec
- fidaxomicin
- finerenone
- fitusiran
- flibanserin
- fluconazole
- fluoxymesterone
- flurbiprofen
- flutamide
- fluticasone
- fluvastatin
- fluvoxamine
- fosamprenavir
- fosaprepitant
- fosinopril
- fosphenytoin
- fostamatinib
- fostemsavir
- fruquintinib
- ganaxolone
- gefitinib
- gemcitabine
- gemfibrozil
- gemtuzumab
- gepirone
- gilteritinib
- givosiran
- glasdegib
- glyburide
- guanfacine
- ibrexafungerp
- ibrutinib
- ibuprofen
- idelalisib
- imatinib
- indacaterol
- indinavir
- indomethacin
- infigratinib
- infliximab
- inotuzumab ozogamicin
- interferon alfa-2a
- interferon alfa-2b
- interferon alfa-n1
- interferon alfacon-1
- interferon beta-1a
- interferon beta-1b
- interferon gamma-1b
- ipilimumab
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isoniazid
- isotretinoin
- istradefylline
- itraconazole
- ivabradine
- ivacaftor
- ixabepilone
- ixazomib
- labetalol
- lamivudine
- lanreotide
- lansoprazole
- lapatinib
- larotrectinib
- lazertinib
- lefamulin
- leflunomide
- lemborexant
- lenacapavir
- lenalidomide
- leniolisib
- lenvatinib
- letermovir
- levobupivacaine
- levofloxacin
- levoketoconazole
- levomethadyl acetate
- levonorgestrel
- lidocaine
- lisinopril
- lomitapide
- lomustine
- lonafarnib
- lonapegsomatropin
- lorlatinib
- lovastatin
- lumateperone
- lurasidone
- lurbinectedin
- lutetium lu 177 dotatate
- macimorelin
- macitentan
- magaldrate
- magnesium carbonate
- magnesium oxide
- maralixibat
- maraviroc
- maribavir
- mavacamten
- mavorixafor
- meclofenamate
- medroxyprogesterone
- mefenamic acid
- mefloquine
- megestrol
- meloxicam
- mephenytoin
- mercaptopurine
- metaxalone
- metformin
- methadone
- methimazole
- methotrexate
- methyldopa
- methylergonovine
- methyltestosterone
- methysergide maleate
- mibefradil
- miconazole
- midostaurin
- mifepristone
- milnacipran
- minocycline
- mipomersen
- mirabegron
- mirikizumab
- mirtazapine
- mitapivat
- mitotane
- mobocertinib
- modafinil
- moexipril
- momelotinib
- mometasone
- monomethyl fumarate
- montelukast
- morphine
- moxifloxacin
- nabumetone
- nafcillin
- naldemedine
- naloxegol
- naltrexone
- nandrolone
- naproxen
- natalizumab
- nefazodone
- nelfinavir
- neratinib
- nevirapine
- niacin
- niacinamide
- nicotinamide
- nifedipine
- nilotinib
- nilutamide
- nintedanib
- niraparib
- nirogacestat
- nitisinone
- nitrofurantoin
- nivolumab
- nizatidine
- norethindrone
- norgestrel
- octreotide
- olaparib
- oliceridine
- olmesartan
- olutasidenib
- omaveloxolone
- omeprazole
- onasemnogene abeparvovec
- oritavancin
- orlistat
- osilodrostat
- osimertinib
- oxaliplatin
- oxandrolone
- oxaprozin
- oxycodone
- oxymetholone
- oxytetracycline
- ozanimod
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palbociclib
- palovarotene
- panobinostat
- pantoprazole
- paricalcitol
- pasireotide
- pazopanib
- pegaspargase
- peginterferon alfa-2a
- peginterferon alfa-2b
- peginterferon beta-1a
- pembrolizumab
- pemigatinib
- pemoline
- pennyroyal
- perampanel
- perindopril
- phenazopyridine
- phenobarbital
- phenylbutazone
- phenytoin
- pimavanserin
- pimecrolimus topical
- pioglitazone
- pirfenidone
- piroxicam
- pirtobrutinib
- pitavastatin
- pitolisant
- polatuzumab vedotin
- pomalidomide
- ponatinib
- ponesimod
- posaconazole
- pralatrexate
- pralsetinib
- pravastatin
- praziquantel
- pretomanid
- primidone
- probenecid
- progesterone
- propylthiouracil
- pyrazinamide
- rabeprazole
- ramelteon
- ramipril
- ranitidine
- ranitidine bismuth citrate
- ranolazine
- red yeast rice
- regorafenib
- relugolix
- remdesivir
- repaglinide
- repotrectinib
- resmetirom
- retapamulin topical
- retifanlimab
- revumenib
- ribociclib
- rifabutin
- rifampin
- rifapentine
- rilpivirine
- riluzole
- rimegepant
- riociguat
- ripretinib
- ritlecitinib
- ritonavir
- rivaroxaban
- rofecoxib
- roflumilast
- rolapitant
- romidepsin
- ropeginterferon alfa-2b
- ropivacaine
- rosiglitazone
- rosuvastatin
- rucaparib
- ruxolitinib
- ruxolitinib topical
- salmeterol
- saquinavir
- sarilumab
- satralizumab
- saxagliptin
- selpercatinib
- selumetinib
- sibutramine
- sildenafil
- silodosin
- simeprevir
- simvastatin
- siponimod
- sirolimus
- sirolimus protein-bound
- sodium bicarbonate
- sodium citrate
- solifenacin
- somapacitan-beco
- somatrem
- somatrogon
- somatropin
- sonidegib
- sorafenib
- sotorasib
- sparsentan
- st. john's wort
- stanozolol
- stavudine
- stiripentol
- sulfadiazine
- sulfadoxine
- sulfamethizole
- sulfamethoxazole
- sulfasalazine
- sulfisoxazole
- sulindac
- sunitinib
- suvorexant
- suzetrigine
- tacrine
- tacrolimus
- tadalafil
- tagraxofusp
- talquetamab
- tamoxifen
- tamsulosin
- tarlatamab
- tasimelteon
- tazemetostat
- teclistamab
- telaprevir
- telithromycin
- telotristat
- temozolomide
- temsirolimus
- teniposide
- tenofovir alafenamide
- tenofovir disoproxil
- tepotinib
- terbinafine
- terfenadine
- teriflunomide
- testosterone
- testosterone topical
- tetracycline
- thioguanine
- thiotepa
- ticagrelor
- tinidazole
- tipranavir
- tislelizumab
- tizanidine
- tocilizumab
- tofacitinib
- tolcapone
- tolmetin
- tolvaptan
- toremifene
- toripalimab
- tovorafenib
- trabectedin
- tramadol
- trandolapril
- tremelimumab
- treosulfan
- tretinoin
- trimetrexate
- trofinetide
- troglitazone
- troleandomycin
- trovafloxacin
- tucatinib
- vadadustat
- valbenazine
- valdecoxib
- valoctocogene roxaparvovec
- valproic acid
- valsartan
- vamorolone
- vandetanib
- vemurafenib
- venetoclax
- venlafaxine
- verapamil
- vibegron
- vilazodone
- viloxazine
- vimseltinib
- vincristine
- vincristine liposome
- vinorelbine
- voclosporin
- vonoprazan
- vorapaxar
- vorasidenib
- voriconazole
- vortioxetine
- voxelotor
- zafirlukast
- zalcitabine
- zaleplon
- zanubrutinib
- zavegepant
- zidovudine
- zileuton
- ziprasidone
- zolpidem
- zonisamide
- zuranolone
Pexidartinib alcohol/food interactions
There are 2 alcohol/food interactions with pexidartinib.
Pexidartinib disease interactions
There are 2 disease interactions with pexidartinib which include:
More about pexidartinib
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- Drug class: multikinase inhibitors
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
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Further information
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