Orladeyo Drug Interactions
Currently displaying a list of 520 drugs known to interact with Orladeyo (berotralstat).
- 79 major drug interactions
- 421 moderate drug interactions
- 20 minor drug interactions
Medications known to interact with Orladeyo
Note: Showing generic names only.
- abemaciclib
- abiraterone
- abrocitinib
- acalabrutinib
- adagrasib
- ado-trastuzumab emtansine
- afatinib
- albendazole
- alfentanil
- alfuzosin
- aliskiren
- alpelisib
- alprazolam
- alvimopan
- ambrisentan
- amiodarone
- amitriptyline
- amlodipine
- amoxapine
- amphetamine
- amprenavir
- apalutamide
- apixaban
- aprepitant
- aripiprazole
- armodafinil
- artesunate
- asciminib
- asenapine
- astemizole
- atazanavir
- atogepant
- atomoxetine
- atorvastatin
- avacopan
- avanafil
- avapritinib
- axitinib
- azelastine nasal
- azelastine ophthalmic
- azithromycin
- bedaquiline
- benzgalantamine
- bepridil
- betamethasone
- betrixaban
- bexarotene
- binimetinib
- bortezomib
- bosentan
- bosutinib
- brentuximab
- brexpiprazole
- brigatinib
- bromocriptine
- budesonide
- budesonide nasal
- buprenorphine
- buspirone
- butorphanol
- cabazitaxel
- cabozantinib
- canagliflozin
- cannabidiol
- cannabis
- capivasertib
- capmatinib
- captopril
- carbamazepine
- cariprazine
- carvedilol
- ceritinib
- cerivastatin
- cevimeline
- chloroquine
- chlorotrianisene
- chlorpheniramine
- chlorpromazine
- cilostazol
- cinacalcet
- cisapride
- citalopram
- cladribine
- clarithromycin
- clindamycin
- clomipramine
- clonazepam
- clopidogrel
- clorazepate
- clozapine
- cobicistat
- cobimetinib
- codeine
- colchicine
- conivaptan
- conjugated estrogens
- cortisone
- crizotinib
- cyclobenzaprine
- cyclophosphamide
- cyclosporine
- dabigatran
- dabrafenib
- daclatasvir
- danicopan
- daridorexant
- darifenacin
- darolutamide
- darunavir
- dasatinib
- daunorubicin
- daunorubicin liposomal
- deflazacort
- delafloxacin
- delavirdine
- desipramine
- deutetrabenazine
- dexamethasone
- dexamethasone nasal
- dexamethasone ophthalmic
- dexfenfluramine
- dexlansoprazole
- dextroamphetamine
- dextromethorphan
- digoxin
- dihydroergotamine
- diltiazem
- diosmiplex
- diphenhydramine
- disopyramide
- docetaxel
- dofetilide
- donepezil
- doravirine
- doxazosin
- doxepin
- doxercalciferol
- doxorubicin
- doxorubicin liposomal
- dronedarone
- droperidol
- drospirenone
- duloxetine
- dutasteride
- duvelisib
- edoxaban
- efavirenz
- elacestrant
- elagolix
- eletriptan
- eliglustat
- eltrombopag
- eluxadoline
- enasidenib
- encorafenib
- enfortumab vedotin
- entrectinib
- enzalutamide
- epirubicin
- eplerenone
- ergonovine
- ergotamine
- erlotinib
- erythromycin
- estazolam
- esterified estrogens
- estradiol
- estradiol topical
- estrone
- estropipate
- estropipate topical
- eszopiclone
- ethinyl estradiol
- ethosuximide
- etonogestrel
- etoposide
- etrasimod
- etravirine
- everolimus
- ezogabine
- febuxostat
- fedratinib
- felodipine
- fenfluramine
- fentanyl
- fesoterodine
- fexinidazole
- fexofenadine
- fidaxomicin
- finerenone
- flecainide
- flibanserin
- fludrocortisone
- flunisolide
- flunisolide nasal
- fluorometholone ophthalmic
- fluoxetine
- fluphenazine
- flurazepam
- fluticasone
- fluticasone nasal
- fluvoxamine
- fosamprenavir
- fosaprepitant
- fostamatinib
- fostemsavir
- fruquintinib
- futibatinib
- halofantrine
- haloperidol
- halothane
- hydrocodone
- hydrocortisone
- hydroxyamphetamine ophthalmic
- hydroxychloroquine
- hydroxyprogesterone
- ibrexafungerp
- ibrutinib
- idarubicin
- idelalisib
- ifosfamide
- iloperidone
- imatinib
- imipramine
- indacaterol
- indinavir
- infigratinib
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isradipine
- istradefylline
- itraconazole
- ivabradine
- ivacaftor
- ivosidenib
- lacosamide
- lapatinib
- larotrectinib
- lasmiditan
- lazertinib
- lemborexant
- lenacapavir
- leniolisib
- letrozole
- levacetylleucine
- levobupivacaine
- levoketoconazole
- levomethadyl acetate
- levonorgestrel
- lidocaine
- lisdexamfetamine
- lomitapide
- lonafarnib
- loperamide
- loratadine
- lorlatinib
- loteprednol ophthalmic
- lovastatin
- lumateperone
- lurasidone
- lusutrombopag
- macitentan
- maprotiline
- maraviroc
- maribavir
- mavacamten
- mavorixafor
- meclizine
- medroxyprogesterone
- mefloquine
- megestrol
- meloxicam
- mesoridazine
- methadone
- methamphetamine
- methotrimeprazine
- methylergonovine
- methylprednisolone
- methysergide maleate
- metoclopramide
- metoprolol
- mexiletine
- mibefradil
- midazolam
- midodrine
- midostaurin
- mifepristone
- mirabegron
- mirtazapine
- mirvetuximab soravtansine
- mitapivat
- mitotane
- mitoxantrone
- mobocertinib
- modafinil
- momelotinib
- mometasone
- mometasone nasal
- mometasone topical
- morphine
- naldemedine
- naloxegol
- naproxen
- nebivolol
- nelfinavir
- neratinib
- nevirapine
- nicardipine
- nifedipine
- nilotinib
- nimodipine
- nintedanib
- niraparib
- nirogacestat
- nisoldipine
- nitisinone
- norethindrone
- norgestrel
- nortriptyline
- olaparib
- oliceridine
- omaveloxolone
- ondansetron
- osilodrostat
- osimertinib
- oteseconazole
- oxybutynin
- oxycodone
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palbociclib
- palovarotene
- panobinostat
- paricalcitol
- paroxetine
- pazopanib
- pemigatinib
- perphenazine
- pexidartinib
- phenytoin
- pimavanserin
- pimecrolimus topical
- pimozide
- pirfenidone
- pirtobrutinib
- pitolisant
- polatuzumab vedotin
- pomalidomide
- ponatinib
- posaconazole
- pralsetinib
- prednisolone
- prednisolone ophthalmic
- prednisone
- pretomanid
- progesterone
- promethazine
- propafenone
- propoxyphene
- propranolol
- protriptyline
- prucalopride
- ramelteon
- ranolazine
- red yeast rice
- regorafenib
- relugolix
- repaglinide
- repotrectinib
- reserpine
- resmetirom
- retapamulin topical
- revumenib
- ribociclib
- rifabutin
- rifampin
- rifapentine
- rilpivirine
- rimegepant
- riociguat
- ripretinib
- risperidone
- ritonavir
- rivaroxaban
- roflumilast
- roflumilast topical
- rolapitant
- romidepsin
- ropivacaine
- rucaparib
- ruxolitinib
- ruxolitinib topical
- safinamide
- salmeterol
- saquinavir
- sarecycline
- saxagliptin
- seladelpar
- selpercatinib
- selumetinib
- sibutramine
- sildenafil
- silodosin
- simeprevir
- simvastatin
- siponimod
- sirolimus
- sirolimus protein-bound
- sirolimus topical
- sofpironium topical
- solifenacin
- sonidegib
- sorafenib
- sotorasib
- sparsentan
- st. john's wort
- stiripentol
- sufentanil
- sunitinib
- suvorexant
- suzetrigine
- tacrolimus
- tadalafil
- tafamidis
- talazoparib
- tamoxifen
- tamsulosin
- tasimelteon
- tazemetostat
- tebentafusp
- tedizolid
- telaprevir
- telithromycin
- temsirolimus
- teniposide
- tenofovir alafenamide
- tenofovir disoproxil
- tepotinib
- terfenadine
- teriflunomide
- testosterone
- tetrabenazine
- thioridazine
- thiotepa
- tiagabine
- ticagrelor
- timolol
- timolol ophthalmic
- tinidazole
- tipranavir
- tisotumab vedotin
- tivozanib
- tofacitinib
- tolterodine
- tolvaptan
- topotecan
- toremifene
- trabectedin
- tramadol
- trazodone
- treosulfan
- tretinoin
- triamcinolone
- triamcinolone nasal
- triamcinolone ophthalmic
- triazolam
- trimipramine
- troglitazone
- troleandomycin
- tucatinib
- vadadustat
- valbenazine
- valdecoxib
- vamorolone
- vandetanib
- vardenafil
- vemurafenib
- venetoclax
- venlafaxine
- verapamil
- vibegron
- vilazodone
- vimseltinib
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- voclosporin
- vorapaxar
- voriconazole
- vortioxetine
- voxelotor
Orladeyo disease interactions
There is 1 disease interaction with Orladeyo (berotralstat) which include:
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- FDA approval history
- Drug class: hereditary angioedema agents
- Breastfeeding
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
See also:
Takhzyro
Takhzyro (lanadelumab-flyo) is used to prevent hereditary angioedema (HAE) and reduce symptoms ...
Berinert
Berinert is used to treat acute abdominal, facial, or laryngeal hereditary angioedema (HAE) attacks ...
Haegarda
Haegarda is an injectable protein replacement therapy that prevents swelling and attacks in ...
Firazyr
Firazyr is used to treat acute attacks of hereditary angioedema (HAE) in adults. It can be ...
Ruconest
Ruconest is used to treat angioedema attacks in adult and adolescent patients with Hereditary ...
Cinryze
Cinryze (complement C1 esterase inhibitor) is used to prevent attacks of angioedema in people with ...
Icatibant
Icatibant is an injection used to treat acute attacks of hereditary angioedema (HAE) in adults. It ...
Lanadelumab
Lanadelumab injection is a monoclonal antibody used to prevent hereditary angioedema. Includes side ...
Stanozolol
Stanozolol is used in the treatment of hereditary angioedema, which causes episodes of swelling of ...
Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.