Efavirenz Drug Interactions
Currently displaying a list of 881 drugs known to interact with efavirenz.
- 276 major drug interactions
- 587 moderate drug interactions
- 18 minor drug interactions
Medications known to interact with efavirenz
Note: Showing generic names only.
- abacavir
- abametapir topical
- abarelix
- abemaciclib
- abiraterone
- abrocitinib
- acalabrutinib
- acarbose
- acetaminophen
- acetylcarbromal
- acitretin
- acoramidis
- acrivastine
- adagrasib
- adalimumab
- adenosine
- ado-trastuzumab emtansine
- afatinib
- albendazole
- albuterol
- aldesleukin
- alectinib
- alefacept
- alfentanil
- alfuzosin
- allopurinol
- almotriptan
- alpelisib
- alprazolam
- amantadine
- ambrisentan
- aminoglutethimide
- aminosalicylic acid
- amiodarone
- amisulpride
- amitriptyline
- amlodipine
- amobarbital
- amoxapine
- amprenavir
- anagrelide
- anakinra
- apixaban
- apomorphine
- apremilast
- aprepitant
- aprocitentan
- arformoterol
- aripiprazole
- armodafinil
- arsenic trioxide
- asciminib
- asenapine
- ashwaganda
- asparaginase erwinia chrysanthemi
- asparaginase escherichia coli
- astemizole
- atazanavir
- atidarsagene autotemcel
- atogepant
- atomoxetine
- atorvastatin
- atovaquone
- atrasentan
- avacopan
- avanafil
- avapritinib
- axitinib
- azatadine
- azithromycin
- baclofen
- baclofen topical
- bedaquiline
- belinostat
- belumosudil
- belzutifan
- benazepril
- benzgalantamine
- bepridil
- berotralstat
- betamethasone
- betibeglogene autotemcel
- bexarotene
- bicalutamide
- bimekizumab
- binimetinib
- bisacodyl
- bitolterol
- black cohosh
- blinatumomab
- boceprevir
- bortezomib
- bosentan
- bosutinib
- brentuximab
- brexanolone
- brexpiprazole
- brigatinib
- brivaracetam
- brodalumab
- bromfenac
- bromocriptine
- brompheniramine
- budesonide
- buprenorphine
- bupropion
- buspirone
- butabarbital
- butalbital
- butorphanol
- cabazitaxel
- cabotegravir
- cabozantinib
- calaspargase pegol
- canakinumab
- cannabidiol
- capivasertib
- capmatinib
- captopril
- carbamazepine
- carbinoxamine
- carfilzomib
- cariprazine
- carisoprodol
- carmustine
- carvedilol
- casanthranol
- cascara sagrada
- caspofungin
- castor oil
- celecoxib
- cenobamate
- ceritinib
- cerivastatin
- cetirizine
- cevimeline
- chaparral
- chenodiol
- chloral hydrate
- chlorcyclizine
- chlordiazepoxide
- chlormezanone
- chloroquine
- chlorotrianisene
- chlorpheniramine
- chlorpromazine
- chlorzoxazone
- cilostazol
- ciprofloxacin
- cisapride
- citalopram
- clarithromycin
- clavulanate
- clemastine
- clobazam
- clofarabine
- clofazimine
- clomipramine
- clonazepam
- clopidogrel
- clorazepate
- clotrimazole
- clozapine
- cobicistat
- cobimetinib
- codeine
- colchicine
- comfrey
- conivaptan
- conjugated estrogens
- conjugated estrogens topical
- copanlisib
- cortisone
- crinecerfont
- crizotinib
- cyclizine
- cyclobenzaprine
- cyclosporine
- cyproheptadine
- cytarabine
- dabrafenib
- dacarbazine
- daclatasvir
- daclizumab
- danazol
- danicopan
- dantrolene
- dapsone
- dapsone topical
- daridorexant
- darifenacin
- darolutamide
- darunavir
- dasatinib
- daunorubicin
- daunorubicin liposomal
- deferasirox
- deflazacort
- degarelix
- dehydroepiandrosterone
- delandistrogene moxeparvovec
- delavirdine
- desipramine
- desloratadine
- desvenlafaxine
- deucravacitinib
- deutetrabenazine
- dexamethasone
- dexbrompheniramine
- dexchlorpheniramine
- dexmedetomidine
- dezocine
- diazepam
- diclofenac
- diclofenac topical
- didanosine
- dienestrol topical
- dihydroergotamine
- diltiazem
- dimenhydrinate
- dimethyl fumarate
- diphenhydramine
- diroximel fumarate
- disopyramide
- disulfiram
- divalproex sodium
- docetaxel
- dofetilide
- dolasetron
- dolutegravir
- donepezil
- doravirine
- doxepin
- doxepin topical
- doxorubicin
- doxorubicin liposomal
- doxylamine
- dronabinol
- dronedarone
- droperidol
- drospirenone
- duloxetine
- dutasteride
- duvelisib
- echinacea
- eflornithine
- elacestrant
- elafibranor
- elagolix
- eletriptan
- eliglustat
- elivaldogene autotemcel
- elotuzumab
- elranatamab
- eltrombopag
- elvitegravir
- emapalumab
- emtricitabine
- enalapril
- enalaprilat
- encorafenib
- enfortumab vedotin
- ensifentrine
- entrectinib
- enzalutamide
- epirubicin
- erdafitinib
- ergonovine
- ergotamine
- eribulin
- erlotinib
- erythromycin
- escitalopram
- esketamine
- estazolam
- esterified estrogens
- estradiol
- estradiol topical
- estrone
- estropipate
- estropipate topical
- eszopiclone
- ethambutol
- ethanol
- ethchlorvynol
- ethinyl estradiol
- ethionamide
- ethosuximide
- ethotoin
- etodolac
- etonogestrel
- etoposide
- etranacogene dezaparvovec
- etrasimod
- etravirine
- etretinate
- everolimus
- exemestane
- ezogabine
- famotidine
- febuxostat
- fedratinib
- felbamate
- felodipine
- fenfluramine
- fenofibrate
- fenofibric acid
- fenoprofen
- fentanyl
- fesoterodine
- fexinidazole
- fexofenadine
- fezolinetant
- fidanacogene elaparvovec
- finerenone
- fingolimod
- fitusiran
- flecainide
- flibanserin
- fluconazole
- fludrocortisone
- fluoxetine
- fluoxymesterone
- fluphenazine
- flurazepam
- flurbiprofen
- flutamide
- fluvastatin
- fluvoxamine
- formoterol
- fosamprenavir
- fosaprepitant
- foscarnet
- fosinopril
- fosphenytoin
- fostamatinib
- fostemsavir
- fruquintinib
- galantamine
- ganaxolone
- gatifloxacin
- gefitinib
- gemcitabine
- gemifloxacin
- gemtuzumab
- gepirone
- gilteritinib
- ginkgo
- givinostat
- givosiran
- glasdegib
- glofitamab
- glycerin
- golimumab
- goserelin
- granisetron
- grepafloxacin
- griseofulvin
- guanfacine
- guselkumab
- halazepam
- halofantrine
- haloperidol
- halothane
- heroin
- histrelin
- hydrocodone
- hydrocortisone
- hydromorphone
- hydroxychloroquine
- hydroxyprogesterone
- hydroxyzine
- ibrexafungerp
- ibrutinib
- ibuprofen
- ibutilide
- idarubicin
- idelalisib
- iloperidone
- imatinib
- imipramine
- indacaterol
- indinavir
- indomethacin
- infigratinib
- infliximab
- inotersen
- inotuzumab ozogamicin
- interferon alfa-2a
- interferon alfa-2b
- interferon alfa-n1
- interferon alfacon-1
- interferon beta-1a
- interferon beta-1b
- interferon gamma-1b
- ipilimumab
- iptacopan
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isocarboxazid
- isoetharine
- isoniazid
- isoproterenol
- isotretinoin
- isradipine
- istradefylline
- itraconazole
- ivabradine
- ivacaftor
- ivermectin
- ivosidenib
- ixabepilone
- ixazomib
- labetalol
- lactitol
- lactulose
- lamivudine
- lapatinib
- larotrectinib
- lazertinib
- lefamulin
- leflunomide
- lemborexant
- lenacapavir
- lenalidomide
- leniolisib
- lenvatinib
- lesinurad
- letermovir
- letrozole
- leuprolide
- levalbuterol
- levamlodipine
- levobupivacaine
- levocetirizine
- levodopa
- levofloxacin
- levoketoconazole
- levomethadyl acetate
- levomilnacipran
- levonorgestrel
- lidocaine
- linagliptin
- lisdexamfetamine
- lisinopril
- lithium
- lofexidine
- lomefloxacin
- lomitapide
- lomustine
- lonafarnib
- lonapegsomatropin
- loperamide
- loratadine
- lorazepam
- lorlatinib
- losartan
- lovastatin
- lovotibeglogene autotemcel
- loxapine
- lumateperone
- lurasidone
- lurbinectedin
- lutetium lu 177 dotatate
- macimorelin
- macitentan
- magnesium citrate
- magnesium hydroxide
- maprotiline
- maralixibat
- maraviroc
- maribavir
- mavacamten
- mavorixafor
- meclizine
- meclofenamate
- medroxyprogesterone
- mefenamic acid
- mefloquine
- megestrol
- melatonin
- meloxicam
- meperidine
- mephenytoin
- mephobarbital
- meprobamate
- mercaptopurine
- mesoridazine
- metaproterenol
- metaxalone
- methadone
- methdilazine
- methimazole
- methocarbamol
- methotrexate
- methotrimeprazine
- methyldopa
- methylergonovine
- methylprednisolone
- methyltestosterone
- methysergide maleate
- metoclopramide
- metronidazole
- mibefradil
- midazolam
- midostaurin
- mifepristone
- milnacipran
- mineral oil
- minocycline
- mipomersen
- mirabegron
- mirikizumab
- mirtazapine
- mitapivat
- mitotane
- mobocertinib
- modafinil
- moexipril
- molindone
- momelotinib
- monomethyl fumarate
- montelukast
- morphine
- morphine liposomal
- moxifloxacin
- nabilone
- nabumetone
- naldemedine
- naloxegol
- naltrexone
- nandrolone
- naproxen
- natalizumab
- nateglinide
- nefazodone
- nelfinavir
- nemolizumab
- neratinib
- nevirapine
- niacin
- niacinamide
- nicardipine
- nicotinamide
- nifedipine
- nilotinib
- nilutamide
- nimodipine
- nintedanib
- nirogacestat
- nisoldipine
- nitisinone
- nitrofurantoin
- norethindrone
- norfloxacin
- norgestrel
- nortriptyline
- ofloxacin
- olanzapine
- olaparib
- oliceridine
- olodaterol
- olutasidenib
- omaveloxolone
- onasemnogene abeparvovec
- ondansetron
- opium
- oritavancin
- orlistat
- orphenadrine
- osilodrostat
- osimertinib
- oxaliplatin
- oxandrolone
- oxaprozin
- oxazepam
- oxcarbazepine
- oxybutynin
- oxycodone
- oxymetholone
- oxymorphone
- oxytocin
- ozanimod
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palbociclib
- paliperidone
- palonosetron
- palovarotene
- panobinostat
- paraldehyde
- paroxetine
- pasireotide
- pazopanib
- pegaspargase
- peginterferon alfa-2a
- peginterferon alfa-2b
- peginterferon beta-1a
- pemigatinib
- pemoline
- pennyroyal
- pentamidine
- pentazocine
- pentobarbital
- perampanel
- perflutren
- perindopril
- perphenazine
- pexidartinib
- phenazopyridine
- phenelzine
- phenindamine
- phenobarbital
- phenolphthalein
- phenylbutazone
- phenytoin
- pimavanserin
- pimozide
- pioglitazone
- pirbuterol
- pirfenidone
- piroxicam
- pirtobrutinib
- pitavastatin
- pitolisant
- polatuzumab vedotin
- polyethylene glycol 3350
- polyethylene glycol 3350 with electrolytes
- ponatinib
- ponesimod
- porfimer
- posaconazole
- pralatrexate
- pralsetinib
- prasugrel
- pravastatin
- praziquantel
- prednisolone
- prednisone
- pretomanid
- primidone
- probucol
- procainamide
- prochlorperazine
- progesterone
- progesterone topical
- proguanil
- promazine
- promethazine
- propafenone
- propofol
- propoxyphene
- propylthiouracil
- protriptyline
- pyrazinamide
- pyrilamine
- rabeprazole
- raltegravir
- ramelteon
- ramipril
- ranolazine
- red yeast rice
- regorafenib
- relugolix
- remdesivir
- remifentanil
- remimazolam
- repaglinide
- repotrectinib
- resmetirom
- revumenib
- ribociclib
- rifabutin
- rifampin
- rifapentine
- rilonacept
- rilpivirine
- riluzole
- rimegepant
- riociguat
- ripretinib
- risperidone
- ritlecitinib
- ritodrine
- ritonavir
- rivaroxaban
- rivastigmine
- rofecoxib
- rolapitant
- romidepsin
- ropeginterferon alfa-2b
- rosiglitazone
- rosuvastatin
- rucaparib
- rufinamide
- ruxolitinib
- ruxolitinib topical
- salmeterol
- saquinavir
- sarilumab
- satralizumab
- saxagliptin
- scopolamine
- secobarbital
- secukinumab
- selpercatinib
- selumetinib
- senna
- sertraline
- sevoflurane
- sildenafil
- silodosin
- siltuximab
- simeprevir
- simvastatin
- siponimod
- sirolimus
- sirolimus protein-bound
- sodium oxybate
- solifenacin
- somapacitan-beco
- somatrem
- somatrogon
- somatropin
- sonidegib
- sorafenib
- sotalol
- sotorasib
- sparfloxacin
- sparsentan
- st. john's wort
- stanozolol
- stavudine
- stiripentol
- sufentanil
- sulfadiazine
- sulfadoxine
- sulfamethizole
- sulfamethoxazole
- sulfasalazine
- sulfinpyrazone
- sulfisoxazole
- sulindac
- sunitinib
- suvorexant
- suzetrigine
- tacrine
- tacrolimus
- tadalafil
- tagraxofusp
- talquetamab
- tamoxifen
- tapentadol
- tarlatamab
- tasimelteon
- tazemetostat
- tebentafusp
- teclistamab
- tecovirimat
- telaprevir
- telavancin
- telithromycin
- telotristat
- temazepam
- temozolomide
- temsirolimus
- teniposide
- tenofovir alafenamide
- tenofovir disoproxil
- tepotinib
- terbinafine
- terbutaline
- terfenadine
- teriflunomide
- testosterone
- testosterone topical
- tetrabenazine
- thalidomide
- thiethylperazine
- thioguanine
- thiopental
- thioridazine
- thiotepa
- thiothixene
- tiagabine
- ticagrelor
- tipranavir
- tizanidine
- tocilizumab
- tofacitinib
- tolcapone
- tolmetin
- tolterodine
- tolvaptan
- toremifene
- torsemide
- tovorafenib
- trabectedin
- tramadol
- trandolapril
- tranylcypromine
- trazodone
- treosulfan
- tretinoin
- triamcinolone
- triazolam
- triclabendazole
- trifluoperazine
- triflupromazine
- trimeprazine
- trimethobenzamide
- trimethoprim
- trimetrexate
- trimipramine
- tripelennamine
- triprolidine
- triptorelin
- trofinetide
- troglitazone
- troleandomycin
- trovafloxacin
- tryptophan
- tucatinib
- vadadustat
- valbenazine
- valdecoxib
- valerian
- valoctocogene roxaparvovec
- valproic acid
- vamorolone
- vandetanib
- vardenafil
- vasopressin
- vemurafenib
- venetoclax
- venlafaxine
- verapamil
- vilazodone
- vimseltinib
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- voclosporin
- vonoprazan
- vorasidenib
- voriconazole
- vortioxetine
- voxelotor
- zafirlukast
- zalcitabine
- zaleplon
- zanubrutinib
- zavegepant
- ziconotide
- zidovudine
- zileuton
- ziprasidone
- zolpidem
- zonisamide
- zuranolone
Efavirenz alcohol/food interactions
There is 1 alcohol/food interaction with efavirenz.
Efavirenz disease interactions
There are 4 disease interactions with efavirenz which include:
More about efavirenz
- efavirenz consumer information
- Check interactions
- Compare alternatives
- Pricing & coupons
- Reviews (8)
- Drug images
- Side effects
- Dosage information
- During pregnancy
- Drug class: NNRTIs
- Breastfeeding
- En español
Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
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Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.