NK1 receptor antagonists
What are NK1 receptor antagonists?
Neurokinin-1 (NK1) receptor antagonists are used for prevention of acute and delayed nausea and vomiting. The NK1 receptor antagonist competitively binds to the NK1 receptor, which blocks the binding of substance P and prevents the emetic signal being transmitted. NK1 receptor antagonists can be used in conjunction with 5-HT3-receptor antagonists and corticosteroids to augment their antiemetic activity.
List of NK1 receptor antagonists
View by Generic | Brand
| Drug Name | Avg. Rating | Reviews |
|---|---|---|
| aprepitant systemic (Pro) Brand names: Emend, Cinvanti, Aponvie |
18 reviews | |
| fosaprepitant systemic (Pro) Brand names: Emend for Injection, Focinvez |
1 review | |
| rolapitant systemic (Pro) Brand name: Varubi |
1 review | |
| For ratings, users were asked how effective they found the medicine while considering positive/adverse effects and ease of use (1 = not effective, 10 = most effective). | ||
See also
Medical conditions treated or associated with NK1 receptor antagonists:
Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.