Tolvaptan Drug Interactions
Currently displaying a list of 354 drugs known to interact with tolvaptan.
- 75 major drug interactions
- 270 moderate drug interactions
- 9 minor drug interactions
Medications known to interact with tolvaptan
Note: Showing generic names only.
- abametapir topical
- abrocitinib
- adagrasib
- adalimumab
- afatinib
- alefacept
- aliskiren
- alpelisib
- amiloride
- aminoglutethimide
- amiodarone
- amobarbital
- amprenavir
- anakinra
- apalutamide
- apixaban
- apomorphine
- aprepitant
- armodafinil
- artesunate
- asciminib
- ashwaganda
- asparaginase erwinia chrysanthemi
- asparaginase escherichia coli
- atazanavir
- avacopan
- azilsartan medoxomil
- bedaquiline
- belzutifan
- benazepril
- bepridil
- berotralstat
- betrixaban
- bexarotene
- bimekizumab
- binimetinib
- black cohosh
- boceprevir
- bosentan
- bosutinib
- brentuximab
- brigatinib
- brodalumab
- butabarbital
- butalbital
- cabozantinib
- calaspargase pegol
- canakinumab
- candesartan
- cannabidiol
- capivasertib
- capmatinib
- captopril
- carbamazepine
- cenobamate
- ceritinib
- chloramphenicol
- ciprofloxacin
- cladribine
- clarithromycin
- clofarabine
- clofazimine
- cobicistat
- cobimetinib
- colchicine
- conivaptan
- crizotinib
- cyclosporine
- dabigatran
- dabrafenib
- daclatasvir
- daclizumab
- danicopan
- daridorexant
- darolutamide
- darunavir
- daunorubicin
- daunorubicin liposomal
- deferasirox
- delafloxacin
- delavirdine
- desmopressin
- dexamethasone
- digoxin
- diltiazem
- docetaxel
- doxorubicin
- doxorubicin liposomal
- dronedarone
- drospirenone
- duvelisib
- echinacea
- edoxaban
- efavirenz
- elacestrant
- elafibranor
- elagolix
- eliglustat
- emapalumab
- empagliflozin
- enalapril
- enalaprilat
- encorafenib
- ensartinib
- enzalutamide
- epirubicin
- eplerenone
- eprosartan
- erdafitinib
- erlotinib
- erythromycin
- etoposide
- etranacogene dezaparvovec
- etravirine
- everolimus
- fedratinib
- felbamate
- fenfluramine
- fexinidazole
- fexofenadine
- fidanacogene elaparvovec
- fidaxomicin
- finerenone
- flibanserin
- fluconazole
- fluvoxamine
- fosamprenavir
- fosaprepitant
- fosinopril
- fosphenytoin
- fostamatinib
- futibatinib
- ibrutinib
- idarubicin
- idelalisib
- imatinib
- indacaterol
- indinavir
- infliximab
- interferon beta-1a
- interferon beta-1b
- iptacopan
- irbesartan
- isavuconazonium
- isoniazid
- istradefylline
- itraconazole
- ivacaftor
- ivosidenib
- lapatinib
- larotrectinib
- lasmiditan
- lazertinib
- lefamulin
- leflunomide
- lenacapavir
- letermovir
- levacetylleucine
- levoketoconazole
- lisinopril
- lomitapide
- lonafarnib
- lonapegsomatropin
- loperamide
- lorlatinib
- losartan
- lovastatin
- lurasidone
- lusutrombopag
- lvp solution with hypertonic saline
- lvp solution with potassium
- maraviroc
- maribavir
- mavacamten
- mavorixafor
- mephobarbital
- methadone
- methotrexate
- metreleptin
- mibefradil
- miconazole
- midostaurin
- mifepristone
- mipomersen
- mitapivat
- mitotane
- mitoxantrone
- mobocertinib
- modafinil
- moexipril
- morphine
- nafcillin
- naldemedine
- naloxegol
- naltrexone
- nefazodone
- nelfinavir
- nemolizumab
- nevirapine
- nifedipine
- nilotinib
- nintedanib
- niraparib
- nirogacestat
- nitisinone
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palovarotene
- parenteral nutrition solution w/electrolytes
- pazopanib
- pegaspargase
- peginterferon beta-1a
- pemigatinib
- pentobarbital
- perindopril
- pexidartinib
- phenobarbital
- phenylbutazone
- phenytoin
- pirtobrutinib
- ponatinib
- posaconazole
- potassium acetate
- potassium acid phosphate
- potassium bicarbonate
- potassium chloride
- potassium citrate
- potassium gluconate
- potassium iodide
- potassium perchlorate
- potassium phosphate
- pralsetinib
- pretomanid
- primidone
- propafenone
- prucalopride
- ramipril
- ranolazine
- relugolix
- remdesivir
- repotrectinib
- ribociclib
- rifabutin
- rifampin
- rifapentine
- rifaximin
- rilonacept
- riociguat
- ripretinib
- ritlecitinib
- ritonavir
- rivaroxaban
- rolapitant
- romidepsin
- rucaparib
- rufinamide
- saquinavir
- sarecycline
- sarilumab
- satralizumab
- secobarbital
- secukinumab
- seladelpar
- selexipag
- selpercatinib
- silodosin
- siltuximab
- sirolimus
- sodium bicarbonate
- sodium chloride
- somapacitan-beco
- somatrem
- somatrogon
- somatropin
- sorafenib
- sotorasib
- sparsentan
- spironolactone
- st. john's wort
- stiripentol
- sulfinpyrazone
- suvorexant
- suzetrigine
- talazoparib
- tamoxifen
- tarlatamab
- teclistamab
- telaprevir
- telithromycin
- telmisartan
- telotristat
- tenofovir alafenamide
- tenofovir disoproxil
- tepotinib
- terfenadine
- teriflunomide
- thioguanine
- ticagrelor
- tipranavir
- tocilizumab
- topotecan
- tovorafenib
- trabectedin
- trandolapril
- treosulfan
- triamterene
- trimethoprim
- trofinetide
- troglitazone
- troleandomycin
- tucatinib
- vadadustat
- valoctocogene roxaparvovec
- valsartan
- vemurafenib
- venetoclax
- verapamil
- vibegron
- viloxazine
- vimseltinib
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- vismodegib
- voclosporin
- vorasidenib
- voriconazole
- voxelotor
Tolvaptan alcohol/food interactions
There is 1 alcohol/food interaction with tolvaptan.
Tolvaptan disease interactions
There are 3 disease interactions with tolvaptan which include:
More about tolvaptan
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- Drug class: vasopressin antagonists
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
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Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.