Ketoconazole Drug Interactions
Currently displaying 404 drugs known to have a major interaction with ketoconazole.
- 404 major drug interactions
- 370 moderate drug interactions
- 39 minor drug interactions
Major interactions with ketoconazole
Note: Showing generic names only.
A
- abacavir
- abemaciclib
- acalabrutinib
- acarbose
- acetaminophen
- acitretin
- adagrasib
- aldesleukin
- alfentanil
- alfuzosin
- alprazolam
- aminosalicylic acid
- amiodarone
- amisulpride
- anagrelide
- apixaban
- arsenic trioxide
- astemizole
- atogepant
- atorvastatin
- atovaquone
- avacopan
- avanafil
- avapritinib
- axitinib
B
- bedaquiline
- belinostat
- belzutifan
- benazepril
- bepridil
- berotralstat
- betrixaban
- blinatumomab
- bosentan
- bosutinib
- brexpiprazole
- brigatinib
- bromfenac
- bromocriptine
- budesonide
- bupropion
- buspirone
- butorphanol
C
- cabozantinib
- capivasertib
- capmatinib
- captopril
- carfilzomib
- cariprazine
- carmustine
- caspofungin
- celecoxib
- ceritinib
- cerivastatin
- chaparral
- chenodeoxycholic acid
- chloroquine
- chlorzoxazone
- cilostazol
- cisapride
- citalopram
- clavulanate
- clotrimazole
- clozapine
- cobimetinib
- colchicine
- comfrey
- conivaptan
- copanlisib
- crizotinib
- cyclosporine
- cytarabine
- cytarabine liposomal
D
- dabigatran
- dacarbazine
- daclatasvir
- danazol
- danicopan
- dantrolene
- daridorexant
- darifenacin
- dasatinib
- deferasirox
- deflazacort
- dehydroepiandrosterone
- delandistrogene moxeparvovec
- demeclocycline
- deucravacitinib
- diclofenac
- diclofenac topical
- dihydroergotamine
- disopyramide
- disulfiram
- divalproex sodium
- docetaxel
- dofetilide
- dolasetron
- doxycycline
- dronedarone
- droperidol
- drospirenone
- duloxetine
- duvelisib
E
- edoxaban
- efavirenz
- eflornithine
- elacestrant
- elagolix
- eletriptan
- eliglustat
- elranatamab
- eltrombopag
- emtricitabine
- enalapril
- enalaprilat
- encorafenib
- enfortumab vedotin
- entrectinib
- eplerenone
- erdafitinib
- ergonovine
- ergotamine
- erythromycin
- escitalopram
- eszopiclone
- ethambutol
- ethionamide
- etodolac
- etranacogene dezaparvovec
- etrasimod
- etretinate
- everolimus
F
- febuxostat
- fedratinib
- felbamate
- felodipine
- fenofibrate
- fenofibric acid
- fenoprofen
- fentanyl
- fesoterodine
- fexinidazole
- fezolinetant
- finerenone
- flibanserin
- fluoxymesterone
- flurbiprofen
- fluticasone
- fluticasone nasal
- fluvastatin
- fosinopril
- fostamatinib
- fruquintinib
- futibatinib
G
H
I
- ibrexafungerp
- ibrutinib
- ibuprofen
- ibutilide
- iloperidone
- indomethacin
- infigratinib
- infliximab
- interferon alfa-2a
- interferon alfa-2b
- interferon alfa-n1
- interferon alfacon-1
- interferon gamma-1b
- ipilimumab
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isotretinoin
- istradefylline
- ivabradine
- ivacaftor
- ivosidenib
K
L
- labetalol
- lamivudine
- lapatinib
- larotrectinib
- lefamulin
- leflunomide
- lemborexant
- lenalidomide
- levoketoconazole
- levomethadyl acetate
- levomilnacipran
- lisinopril
- lomitapide
- lomustine
- lonafarnib
- loperamide
- lorlatinib
- lovastatin
- lumateperone
- lurasidone
- lurbinectedin
M
- macitentan
- maraviroc
- mavacamten
- meclofenamate
- mefenamic acid
- mefloquine
- meloxicam
- mercaptopurine
- mesoridazine
- metaxalone
- methadone
- methimazole
- methyldopa
- methylergonovine
- methylprednisolone
- methyltestosterone
- methysergide maleate
- midazolam
- midostaurin
- mifepristone
- milnacipran
- minocycline
- mipomersen
- mirikizumab
- mirvetuximab soravtansine
- mitapivat
- mobocertinib
- moexipril
- momelotinib
- morphine
- moxifloxacin
N
- nabumetone
- naloxegol
- nandrolone
- naproxen
- natalizumab
- neratinib
- niacin
- niacinamide
- nilotinib
- nimodipine
- nirogacestat
- nisoldipine
- nitrofurantoin
O
- olaparib
- oliceridine
- onasemnogene abeparvovec
- orlistat
- osilodrostat
- osimertinib
- oxandrolone
- oxaprozin
- oxycodone
- oxymetholone
- oxytetracycline
- ozanimod
P
- pacritinib
- palbociclib
- palovarotene
- panobinostat
- papaverine
- pasireotide
- pazopanib
- peginterferon alfa-2a
- peginterferon alfa-2b
- pemigatinib
- pemoline
- pennyroyal
- perindopril
- pexidartinib
- phenazopyridine
- phenylbutazone
- pimavanserin
- pimozide
- pirfenidone
- piroxicam
- pirtobrutinib
- pitavastatin
- polatuzumab vedotin
- ponatinib
- ponesimod
- posaconazole
- pralatrexate
- pralsetinib
- pravastatin
- procainamide
- propylthiouracil
- pyrazinamide
Q
R
- ramipril
- ranolazine
- red yeast rice
- relugolix
- repotrectinib
- resmetirom
- ribociclib
- rifabutin
- rifampin
- rifapentine
- riluzole
- rimegepant
- riociguat
- ripretinib
- ritonavir
- rivaroxaban
- rofecoxib
- ropeginterferon alfa-2b
- rosuvastatin
- ruxolitinib
S
- salmeterol
- selpercatinib
- selumetinib
- sildenafil
- silodosin
- simeprevir
- simvastatin
- siponimod
- sirolimus
- sirolimus protein-bound
- solifenacin
- sonidegib
- sotalol
- sparfloxacin
- sparsentan
- stanozolol
- stavudine
- sulfadiazine
- sulfadoxine
- sulfamethizole
- sulfasalazine
- sulfisoxazole
- sulindac
- suvorexant
T
- tacrolimus
- tadalafil
- talquetamab
- tamsulosin
- tazemetostat
- teclistamab
- telithromycin
- temozolomide
- temsirolimus
- tenofovir
- tenofovir alafenamide
- tepotinib
- terfenadine
- teriflunomide
- testosterone
- testosterone topical
- tetracycline
- thioridazine
- ticagrelor
- tisotumab vedotin
- tocilizumab
- tofacitinib
- tolcapone
- tolmetin
- tolvaptan
- toremifene
- trabectedin
- trandolapril
- tretinoin
- triamcinolone
- triazolam
- troglitazone
- troleandomycin
- trovafloxacin
U
V
- valbenazine
- valproic acid
- vandetanib
- vardenafil
- vemurafenib
- venetoclax
- vilazodone
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- voclosporin
- vorapaxar
- voxelotor
Z
Ketoconazole alcohol/food interactions
There is 1 alcohol/food interaction with ketoconazole.
Ketoconazole disease interactions
There are 4 disease interactions with ketoconazole which include:
More about ketoconazole
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.