Ketoconazole Drug Interactions
Currently displaying a list of 854 drugs known to interact with ketoconazole.
- 431 major drug interactions
- 384 moderate drug interactions
- 39 minor drug interactions
Medications known to interact with ketoconazole
Note: Showing generic names only.
A
- abacavir
- abametapir topical
- abarelix
- abemaciclib
- abiraterone
- abrocitinib
- acalabrutinib
- acarbose
- acetaminophen
- acitretin
- adagrasib
- adenosine
- ado-trastuzumab emtansine
- afatinib
- albuterol
- aldesleukin
- alfentanil
- alfuzosin
- aliskiren
- allopurinol
- almotriptan
- alosetron
- alprazolam
- aluminum carbonate
- aluminum hydroxide
- ambrisentan
- aminophylline
- aminosalicylic acid
- amiodarone
- amisulpride
- amitriptyline
- amlodipine
- amoxapine
- amphotericin b
- amphotericin b cholesteryl sulfate
- amphotericin b lipid complex
- amphotericin b liposomal
- amprenavir
- anagrelide
- anisindione
- apalutamide
- apixaban
- apomorphine
- aprepitant
- aprocitentan
- arformoterol
- aripiprazole
- armodafinil
- arsenic trioxide
- asciminib
- asenapine
- ashwaganda
- asparaginase erwinia chrysanthemi
- asparaginase escherichia coli
- astemizole
- atazanavir
- atezolizumab
- atogepant
- atomoxetine
- atorvastatin
- atovaquone
- atrasentan
- atropine
- avacopan
- avanafil
- avapritinib
- avatrombopag
- avelumab
- axitinib
- azithromycin
B
- bedaquiline
- belinostat
- belladonna
- belumosudil
- belzutifan
- benazepril
- benzgalantamine
- benztropine
- bepridil
- berotralstat
- betamethasone
- betrixaban
- bexarotene
- bicalutamide
- binimetinib
- biperiden
- bisacodyl
- bitolterol
- black cohosh
- blinatumomab
- boceprevir
- bortezomib
- bosentan
- bosutinib
- brentuximab
- brewer's yeast
- brexpiprazole
- brigatinib
- brivaracetam
- bromfenac
- bromocriptine
- budesonide
- budesonide nasal
- buprenorphine
- bupropion
- buspirone
- busulfan
- butorphanol
C
- cabazitaxel
- cabozantinib
- calaspargase pegol
- calcium carbonate
- cannabidiol
- cannabis
- capivasertib
- capmatinib
- captopril
- carbamazepine
- carfilzomib
- cariprazine
- carmustine
- casanthranol
- cascara sagrada
- caspofungin
- castor oil
- celecoxib
- cemiplimab
- cenobamate
- ceritinib
- cerivastatin
- cevimeline
- chaparral
- chenodiol
- chloroquine
- chlorotrianisene
- chlorpromazine
- chlorzoxazone
- ciclesonide
- ciclesonide nasal
- cilostazol
- cimetidine
- cinacalcet
- ciprofloxacin
- cisapride
- citalopram
- clarithromycin
- clavulanate
- clidinium
- clindamycin
- clobazam
- clofarabine
- clofazimine
- clomipramine
- clopidogrel
- clotrimazole
- clozapine
- cobicistat
- cobimetinib
- coccidioidin skin test
- colchicine
- comfrey
- conivaptan
- conjugated estrogens
- conjugated estrogens topical
- copanlisib
- cortisone
- cosibelimab
- crizotinib
- cyclosporine
- cytarabine
- cytarabine liposomal
D
- dabigatran
- dabrafenib
- dacarbazine
- daclatasvir
- daclizumab
- dalfampridine
- danazol
- danicopan
- dantrolene
- daprodustat
- daridorexant
- darifenacin
- darolutamide
- darunavir
- dasatinib
- daunorubicin
- daunorubicin liposomal
- deferasirox
- deflazacort
- degarelix
- dehydroepiandrosterone
- delandistrogene moxeparvovec
- delavirdine
- demeclocycline
- desipramine
- desloratadine
- deucravacitinib
- deutetrabenazine
- dexamethasone
- dexamethasone nasal
- dexamethasone ophthalmic
- dexlansoprazole
- diazepam
- diclofenac
- diclofenac topical
- dicumarol
- dicyclomine
- didanosine
- dienestrol topical
- diethylstilbestrol
- digoxin
- dihydroergotamine
- dihydroxyaluminum sodium carbonate
- diltiazem
- dimethyl fumarate
- diroximel fumarate
- disopyramide
- disulfiram
- divalproex sodium
- docetaxel
- dofetilide
- dolasetron
- dolutegravir
- donepezil
- doravirine
- dostarlimab
- doxazosin
- doxepin
- doxorubicin
- doxorubicin liposomal
- doxycycline
- dronedarone
- droperidol
- drospirenone
- duloxetine
- durvalumab
- dutasteride
- duvelisib
E
- echinacea
- edoxaban
- efavirenz
- eflornithine
- elacestrant
- elagolix
- eletriptan
- eliglustat
- elranatamab
- eltrombopag
- eluxadoline
- emtricitabine
- enalapril
- enalaprilat
- encorafenib
- enfortumab vedotin
- entrectinib
- enzalutamide
- epirubicin
- eplerenone
- eravacycline
- erdafitinib
- ergonovine
- ergotamine
- eribulin
- erlotinib
- erythromycin
- escitalopram
- esomeprazole
- esterified estrogens
- estradiol
- estradiol topical
- estrone
- estropipate
- estropipate topical
- eszopiclone
- ethambutol
- ethanol
- ethinyl estradiol
- ethionamide
- ethotoin
- etodolac
- etonogestrel
- etranacogene dezaparvovec
- etrasimod
- etravirine
- etretinate
- everolimus
- ezogabine
F
- famotidine
- febuxostat
- fedratinib
- felbamate
- felodipine
- fenfluramine
- fenofibrate
- fenofibric acid
- fenoprofen
- fentanyl
- fesoterodine
- fexinidazole
- fexofenadine
- fezolinetant
- fidanacogene elaparvovec
- fidaxomicin
- finerenone
- fingolimod
- fitusiran
- flavoxate
- flecainide
- flibanserin
- flotufolastat F 18
- fluconazole
- fludrocortisone
- flunisolide
- flunisolide nasal
- fluorometholone ophthalmic
- fluoxetine
- fluoxymesterone
- fluphenazine
- flurbiprofen
- flutamide
- fluticasone
- fluticasone nasal
- fluvastatin
- fluvoxamine
- formoterol
- fosamprenavir
- fosaprepitant
- foscarnet
- fosinopril
- fosphenytoin
- fostamatinib
- fostemsavir
- fruquintinib
- futibatinib
G
- galantamine
- gallium Ga 68 gozetotide
- gallium ga 68 psma-11
- ganaxolone
- gatifloxacin
- gefitinib
- gemcitabine
- gemifloxacin
- gemtuzumab
- gepirone
- gilteritinib
- givinostat
- glasdegib
- glycerin
- glycopyrrolate
- goserelin
- granisetron
- grepafloxacin
- griseofulvin
- guanfacine
H
- halofantrine
- haloperidol
- halothane
- histrelin
- hydrocodone
- hydrocortisone
- hydroxychloroquine
- hydroxyprogesterone
- hydroxyzine
- hyoscyamine
I
- ibrexafungerp
- ibrutinib
- ibuprofen
- ibutilide
- idarubicin
- idelalisib
- iloperidone
- imatinib
- imipramine
- indacaterol
- indinavir
- indomethacin
- infigratinib
- infliximab
- inotuzumab ozogamicin
- interferon alfa-2a
- interferon alfa-2b
- interferon alfa-n1
- interferon alfacon-1
- interferon beta-1a
- interferon beta-1b
- interferon gamma-1b
- ipilimumab
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isoetharine
- isoniazid
- isoproterenol
- isotretinoin
- isradipine
- istradefylline
- ivabradine
- ivacaftor
- ivermectin
- ivosidenib
- ixabepilone
K
L
- labetalol
- lacosamide
- lactitol
- lactulose
- lamivudine
- lansoprazole
- lanthanum carbonate
- lapatinib
- larotrectinib
- lazertinib
- lefamulin
- leflunomide
- lemborexant
- lenacapavir
- lenalidomide
- leniolisib
- lenvatinib
- leuprolide
- levalbuterol
- levamlodipine
- levobupivacaine
- levofloxacin
- levoketoconazole
- levomethadyl acetate
- levomilnacipran
- levonorgestrel
- lidocaine
- lisdexamfetamine
- lisinopril
- lithium
- lofexidine
- lomefloxacin
- lomitapide
- lomustine
- lonafarnib
- lonapegsomatropin
- loperamide
- loratadine
- lorlatinib
- losartan
- loteprednol ophthalmic
- lovastatin
- lumateperone
- lurasidone
- lurbinectedin
- lusutrombopag
M
- macimorelin
- macitentan
- magaldrate
- magnesium carbonate
- magnesium citrate
- magnesium hydroxide
- magnesium oxide
- maprotiline
- maralixibat
- maraviroc
- mavacamten
- mavorixafor
- meclofenamate
- medroxyprogesterone
- mefenamic acid
- mefloquine
- megestrol
- meloxicam
- mepenzolate
- mephenytoin
- mercaptopurine
- mesoridazine
- metaproterenol
- metaxalone
- methadone
- methimazole
- methotrexate
- methotrimeprazine
- methscopolamine
- methyldopa
- methylergonovine
- methylprednisolone
- methyltestosterone
- methysergide maleate
- metronidazole
- mibefradil
- midazolam
- midostaurin
- mifepristone
- milnacipran
- mineral oil
- minocycline
- mipomersen
- mirabegron
- mirikizumab
- mirtazapine
- mirvetuximab soravtansine
- mitapivat
- mitotane
- mitoxantrone
- mobocertinib
- modafinil
- moexipril
- momelotinib
- mometasone
- mometasone nasal
- monomethyl fumarate
- morphine
- moxifloxacin
N
- nabumetone
- naldemedine
- naloxegol
- naltrexone
- nandrolone
- naproxen
- natalizumab
- nefazodone
- nelfinavir
- neratinib
- nevirapine
- niacin
- niacinamide
- nicardipine
- nicotinamide
- nifedipine
- nilotinib
- nilutamide
- nimodipine
- nintedanib
- niraparib
- nirogacestat
- nisoldipine
- nitisinone
- nitrofurantoin
- nivolumab
- nizatidine
- norethindrone
- norfloxacin
- norgestrel
- nortriptyline
O
- obeticholic acid
- ofloxacin
- olanzapine
- olaparib
- oliceridine
- olodaterol
- olutasidenib
- omaveloxolone
- omeprazole
- onasemnogene abeparvovec
- ondansetron
- orlistat
- osilodrostat
- osimertinib
- ospemifene
- oxaliplatin
- oxandrolone
- oxaprozin
- oxcarbazepine
- oxtriphylline
- oxybutynin
- oxycodone
- oxymetholone
- oxytetracycline
- oxytocin
- ozanimod
P
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palbociclib
- paliperidone
- palonosetron
- palovarotene
- panobinostat
- pantoprazole
- papaverine
- paricalcitol
- pasireotide
- pazopanib
- pegaspargase
- peginterferon alfa-2a
- peginterferon alfa-2b
- peginterferon beta-1a
- pembrolizumab
- pemigatinib
- pemoline
- pennyroyal
- pentamidine
- perampanel
- perflutren
- perindopril
- perphenazine
- pexidartinib
- phenazopyridine
- phenobarbital
- phenolphthalein
- phenylbutazone
- phenytoin
- piflufolastat F 18
- pimavanserin
- pimecrolimus topical
- pimozide
- pioglitazone
- pirbuterol
- pirfenidone
- piroxicam
- pirtobrutinib
- pitavastatin
- pitolisant
- polatuzumab vedotin
- polyethylene glycol 3350
- polyethylene glycol 3350 with electrolytes
- pomalidomide
- ponatinib
- ponesimod
- porfimer
- posaconazole
- pralatrexate
- pralsetinib
- pravastatin
- prednisolone
- prednisolone ophthalmic
- prednisone
- primaquine
- primidone
- probucol
- procainamide
- prochlorperazine
- procyclidine
- progesterone
- progesterone topical
- promazine
- promethazine
- propafenone
- propantheline
- propofol
- propoxyphene
- propylthiouracil
- protriptyline
- prucalopride
- pyrazinamide
Q
R
- rabeprazole
- ramelteon
- ramipril
- ranitidine
- ranitidine bismuth citrate
- ranolazine
- red yeast rice
- regorafenib
- relugolix
- remdesivir
- repaglinide
- repotrectinib
- resmetirom
- retapamulin topical
- retifanlimab
- revumenib
- ribociclib
- rifabutin
- rifampin
- rifapentine
- rilpivirine
- riluzole
- rimegepant
- riociguat
- ripretinib
- risperidone
- ritlecitinib
- ritodrine
- ritonavir
- rivaroxaban
- rivastigmine
- rofecoxib
- roflumilast
- roflumilast topical
- romidepsin
- ropeginterferon alfa-2b
- ropivacaine
- rosiglitazone
- rosuvastatin
- rucaparib
- ruxolitinib
- ruxolitinib topical
S
- saccharomyces boulardii lyo
- salmeterol
- saquinavir
- saxagliptin
- scopolamine
- seladelpar
- selpercatinib
- selumetinib
- senna
- sertraline
- sevoflurane
- sibutramine
- sildenafil
- silodosin
- simeprevir
- simvastatin
- siponimod
- sirolimus
- sirolimus protein-bound
- sirolimus topical
- sodium bicarbonate
- sodium zirconium cyclosilicate
- solifenacin
- somapacitan-beco
- somatrem
- somatrogon
- somatropin
- sonidegib
- sorafenib
- sotalol
- sotorasib
- sparfloxacin
- sparsentan
- st. john's wort
- stanozolol
- stavudine
- stiripentol
- sucralfate
- sufentanil
- sulfadiazine
- sulfadoxine
- sulfamethizole
- sulfamethoxazole
- sulfasalazine
- sulfisoxazole
- sulindac
- sunitinib
- suvorexant
- suzetrigine
T
- tacrine
- tacrolimus
- tadalafil
- talazoparib
- talquetamab
- tamoxifen
- tamsulosin
- tarlatamab
- tasimelteon
- tazemetostat
- tebentafusp
- teclistamab
- tecovirimat
- telaprevir
- telavancin
- telithromycin
- telotristat
- temozolomide
- temsirolimus
- tenofovir alafenamide
- tenofovir disoproxil
- tepotinib
- terbinafine
- terbutaline
- terfenadine
- teriflunomide
- testosterone
- testosterone topical
- tetrabenazine
- tetracycline
- thalidomide
- theophylline
- thioguanine
- thioridazine
- thiotepa
- ticagrelor
- tipranavir
- tislelizumab
- tisotumab vedotin
- tizanidine
- tocilizumab
- tofacitinib
- tolbutamide
- tolcapone
- tolmetin
- tolterodine
- tolvaptan
- toremifene
- toripalimab
- tovorafenib
- trabectedin
- tramadol
- trandolapril
- trazodone
- tremelimumab
- treosulfan
- tretinoin
- triamcinolone
- triamcinolone nasal
- triamcinolone ophthalmic
- triazolam
- triclabendazole
- trifluoperazine
- triflupromazine
- trihexyphenidyl
- trimeprazine
- trimetrexate
- trimipramine
- triptorelin
- trofinetide
- troglitazone
- troleandomycin
- trospium
- trovafloxacin
- tucatinib
U
V
- vadadustat
- valbenazine
- valdecoxib
- valoctocogene roxaparvovec
- valproic acid
- vamorolone
- vandetanib
- vardenafil
- vasopressin
- vemurafenib
- venetoclax
- venlafaxine
- verapamil
- vilazodone
- vimseltinib
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- vismodegib
- voclosporin
- vonoprazan
- vorapaxar
- vorasidenib
- voriconazole
- voxelotor
W
Z
- zafirlukast
- zalcitabine
- zanubrutinib
- zavegepant
- zidovudine
- zileuton
- ziprasidone
- zolpidem
- zonisamide
- zuranolone
Ketoconazole alcohol/food interactions
There is 1 alcohol/food interaction with ketoconazole.
Ketoconazole disease interactions
There are 4 disease interactions with ketoconazole which include:
More about ketoconazole
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.