Tacrolimus
In some countries, this medicine may only be approved for veterinary use.
In the US, Tacrolimus (tacrolimus systemic) is a member of the drug class calcineurin inhibitors and is used to treat Crohn's Disease, Graft-versus-host disease, Organ Transplant - Rejection Prophylaxis and Organ Transplant - Rejection Reversal.
US matches:
- Tacrolimus
- Tacrolimus capsules
- Tacrolimus ointment
- Tacrolimus oral and injection
- Tacrolimus topical
- Tacrolimus Intravenous
- Tacrolimus Oral, Intravenous
Scheme
Rec.INN
ATC (Anatomical Therapeutic Chemical Classification)
D11AH01,L04AA05,L04AD02
CAS registry number (Chemical Abstracts Service)
0104987-11-3
Chemical Formula
C44-H69-N-O12
Molecular Weight
804
Therapeutic Category
Immunosuppressant
Chemical Name
Immunosuppressant derived from Streptomyces tsukubaensis
Foreign Names
- Tacrolimusum (Latin)
- Tacrolimus (German)
- Tacrolimus (French)
- Tacrolimus (Spanish)
Generic Names
- Tacrolimus (OS: USAN, BAN)
- Tacrolimus Hydrate (OS: JAN)
- FK 506 (IS: Fujisawa)
- FR 900506 (IS)
- L 683590 (IS)
- Tacrolimus Hydrate (PH: JP XV)
Brand Names
- Advagraf
Astellas, Belgium; Astellas, Canada; Astellas, China; Astellas, Czech Republic; Astellas, Denmark; Astellas, Georgia; Astellas, Greece; Astellas, Hong Kong; Astellas, Hungary; Astellas, Iceland; Astellas, Netherlands; Astellas, Norway; Astellas, Poland; Astellas, Portugal; Astellas, Romania; Astellas, Slovakia; Astellas, Taiwan; Astellas Pharma, Switzerland; Astellas Pharma, Spain; Astellas Pharma, Italy; Astellas Pharma, Latvia; Astellas Pharma GmbH, Luxembourg; PharmaSwiss, Croatia (Hrvatska) - Aristoderm
Ariston, Argentina - Atolimus
Beximco, Bangladesh - Capexion (veterinary use)
Mylan, United Kingdom - Crolim
Ranbaxy, India - Cromidin
Royal Pharma, Chile - Effac
Meider, Taiwan - Modigraf
Astellas, Lithuania - Mustopic
Systopic, India - Proalid
Darier, Mexico - Prograf
Al Hikma, Oman; Astellas, Austria; Astellas, Bosnia & Herzegowina; Astellas, Canada; Astellas, China; Astellas, Czech Republic; Astellas, Germany; Astellas, Denmark; Astellas, Finland; Astellas, Georgia; Astellas, Greece; Astellas, Hong Kong; Astellas, Hungary; Astellas, Indonesia; Astellas, Ireland; Astellas, Israel; Astellas, Iceland; Astellas, South Korea; Astellas, Norway; Astellas, Philippines; Astellas, Poland; Astellas, Portugal; Astellas, Romania; Astellas, Russian Federation; Astellas, Slovakia; Astellas, Thailand; Astellas, Turkey; Astellas, Taiwan; Astellas, United States; Astellas, Vietnam; Astellas, South Africa; Astellas Pharma, Switzerland; Astellas Pharma, Spain; Astellas Pharma, Italy; Astellas Pharma, Sweden; Gador, Argentina; Hikma, Tunisia; Janssen, Brazil; Janssen, Malaysia; Janssen, New Zealand; Janssen, Venezuela; Janssen-Cilag, Singapore; Pharma Investi, Chile; PharmaSwiss, Slovenia - Prograft
Astellas, Belgium; Astellas, Netherlands; Astellas Pharma S.A., Luxembourg - Protopic
Astellas, Canada; Astellas, China; Astellas, Georgia; Astellas, Greece; Astellas, Hong Kong; Astellas, Indonesia; Astellas, Lithuania; Astellas, Norway; Astellas, Romania; Astellas, Turkey; Astellas, Taiwan; Astellas, United States; Astellas Pharma, Switzerland; Astellas Pharma, Spain; Astellas Pharma, Latvia; Astellas/ Janssen-Cilag, Vietnam; Janssen, Malaysia; Janssen, Philippines; Janssen-Cilag, Indonesia; Janssen-Cilag, Singapore; Roche, Peru; Roche, Uruguay; Roche, Venezuela - Protopy
Fujisawa, Latvia - Remus
Square, Bangladesh - Seegraf
Micro Labs, India - Susciter
Aversi, Georgia - Tacni
Teva, Bulgaria; Teva, Estonia; Teva, Sweden; Teva Pharmaceuticals, United Kingdom - Tacroderm
Abbott, India - Tacrograf
Biocon, India - Tacrokid (pediatric)
Elder, India - Tacrol
Acme, Bangladesh - Tacroli
Hwang's, Taiwan - Tacrolim
Incepta, Bangladesh - Tacrolimus Accord
Accord Healthcare, United States - Tacrolimus Actavis
Actavis, Switzerland - Tacrolimus Dr. Reddy's
Dr. Reddy's, United States - Tacrolimus Intas
Accord Healthcare, Estonia - Tacrolimus Lek
Sandoz, Georgia - Tacrolimus Mylan
Mylan, United States - Tacrolimus Sandoz
Sandoz, Switzerland; Sandoz, United States - Tacrolimus Watson
Watson, United States - Tacrolimus
Accord Healthcare, Malta - Tacrolimus-Teva
Teva Pharma, Switzerland - Tacromus
Zydus Cadila, India - Tacroz
Glenmark, India; Glenmark, Vietnam - Tagraf
Panacea Biotech, Philippines - Takon
Arrow, Malta - Taliximun
Cinfa, Bulgaria - T-Inmun
Biomedical, Chile; Mediderm, Chile; Mediderm, Peru - Traderma
Serral, Mexico - Vingraf
Emcure Pharma, Philippines - Adoport
Sandoz, United Kingdom - Advagraf
Astellas, Germany; Astellas, Finland; Astellas, France; Astellas, United Kingdom; Astellas, Ireland; Astellas, Lithuania; Astellas Pharma, Sweden; Astellas Pharma Europe, Austria - Framebin
Pisa, Mexico - Graceptor
Astellas Pharma, Japan - Limustin
Landsteiner, Mexico - Modigraf
Astellas, Germany; Astellas, France; Astellas, United Kingdom; Astellas Pharma, Latvia; Astellas Pharma, Sweden - Pangraf
Panacea, Georgia - Prograf
Astellas, Austria; Astellas, Bulgaria; Astellas, France; Astellas, United Kingdom; Astellas, Malta; Astellas, Serbia; Astellas Pharma, Japan; Astellas Pharma, Sweden; Janssen-Cilag, Colombia; P & D, Malta; PharmaSwiss, Croatia (Hrvatska) - Prograft
Astellas, Netherlands - Protopic
Al Hikma, Oman; Astellas, Belgium; Astellas, Czech Republic; Astellas, Germany; Astellas, Denmark; Astellas, Finland; Astellas, France; Astellas, United Kingdom; Astellas, Hungary; Astellas, Ireland; Astellas, Israel; Astellas, Iceland; Astellas, South Korea; Astellas, Netherlands; Astellas, Poland; Astellas, Portugal; Astellas, South Africa; Astellas Pharma, Italy; Astellas Pharma, Japan; Astellas Pharma, Sweden; Astellas Pharma Europe, Austria; Fujisawa, Slovenia; Fujisawa, Slovakia; Janssen, Thailand; Roche, Argentina; Roche, Chile; Roche, Colombia; Roche, Ecuador; Roche, Mexico - Tacrobell
Chong Kun Dang, South Korea - Tacrocel
Sandoz, Croatia (Hrvatska) - Tacrocin
Intas, Philippines - Tacrolimus Hexal
Hexal, Germany - Tacrolimus Sandoz
Sandoz, Austria; Sandoz, Australia; Sandoz, Sweden - Talymus
Senju Seiyaku, Japan
International Drug Name Search
Glossary
| Term | Definition |
|---|---|
| BAN | British Approved Name |
| IS | Inofficial Synonym |
| JAN | Japanese Accepted Name |
| OS | Official Synonym |
| PH | Pharmacopoeia Name |
| Rec.INN | Recommended International Nonproprietary Name (World Health Organization) |
| USAN | United States Adopted Name |
Click for further information on drug naming conventions and International Nonproprietary Names.
Important Notice: The Drugs.com international database is in BETA release. This means it is still under development and may contain inaccuracies. It is not intended as a substitute for the expertise and judgement of your physician, pharmacist or other healthcare professional. It should not be construed to indicate that the use of any medication in any country is safe, appropriate or effective for you. Consult with your healthcare professional before taking any medication.


