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Raltegravir

In the US, Raltegravir (raltegravir systemic) is a member of the drug class integrase strand transfer inhibitor and is used to treat HIV Infection and Occupational Exposure.

US matches:

Scheme

Rec.INN

ATC (Anatomical Therapeutic Chemical Classification)

J05AX08

CAS registry number (Chemical Abstracts Service)

0518048-05-0

Chemical Formula

C20-H21-F-N6-O5

Molecular Weight

444

Therapeutic Categories

Antivirals for systemic use - Antiviral agent

Treatment of HIV infection

HIV integrase inhibitor

Chemical Names

N-[(4-Fluorophenyl)metyl]-5-hydroxy-1-metyl-2-[2-(5-metyl-1,3,4-oxadiazole-2-carboxamido)propan-2-yl]-6-oxo-1,6-dihydropyrimidine-4-carboxamide (WHO)

4-Pyrimidinecarboxamide, N-((4-fluorophenyl)metyl)-1,6-dihydro-5-hydroxy-1-metyl-2-(1-metyl-1-(((5-metyl-1,3,4-oxadiazol-2-yl)carbonyl)amino)etyl)-6-oxo-

5-Hydroxy-1-metyl-2-{1-metyl-1-[(5-metyl[1,3,4]oxadiazol-2-carbonyl)amino]etyl}-6-oxo-1,6-dihydropyrimidin-4-carbonsäure-4-fluorbenzylamid (IUPAC)

N-(2-(4-(4-Fluorobenzylcarbamoyl)-5-hydroxy-1-metyl-6-oxo-1,6-dihydropyrimidin-2-yl)propan-2-yl)-5-metyl-1,3,4-oxadiazole-2-carboxamide

Foreign Names

  • Raltegravirum (Latin)
  • Raltegravir (German)
  • Raltégravir (French)
  • Raltegravir (Spanish)

Generic Names

Brand Names

  • Dutrebis [+ Lamivudine]
    Merck Sharp & Dohme, Lithuania; Merck Sharp & Dohme, Poland
  • Isentress
    Cibeles, Uruguay; Merck, Turkey; Merck Sharp & Dohme, Cyprus; Merck Sharp & Dohme, Greece; Merck Sharp & Dohme, Hong Kong; Merck Sharp & Dohme, Malaysia; Merck Sharp & Dohme, Netherlands; Merck Sharp & Dohme, Slovenia; Merck Sharp & Dohme, Taiwan; MSD, Costa Rica; MSD, Dominican Republic; MSD, Guatemala; MSD, Honduras; MSD, Nicaragua; MSD, Panama; MSD, Slovakia; MSD, El Salvador; MSD, Thailand; MSD, South Africa; MSD Italia, Italy; Merck Sharp & Dohme Pharma Singapore, Singapore
  • Dutrebis [+ Lamivudine]
    Merck Sharp & Dohme, United States
  • Isentress
    Merck Canada, Canada; Merck Sharp & Dohme, Australia; Merck Sharp & Dohme, Bosnia & Herzegowina; Merck Sharp & Dohme, Brazil; Merck Sharp & Dohme, Chile; Merck Sharp & Dohme, Estonia; Merck Sharp & Dohme, Spain; Merck Sharp & Dohme, United Kingdom; Merck Sharp & Dohme, Georgia; Merck Sharp & Dohme, Croatia (Hrvatska); Merck Sharp & Dohme, Iceland; Merck Sharp & Dohme, Lithuania; Merck Sharp & Dohme, Latvia; Merck Sharp & Dohme, New Zealand; Merck Sharp & Dohme, Poland; Merck Sharp & Dohme, Romania; Merck Sharp & Dohme, Serbia; Merck Sharp & Dohme, United States; MSD, Czech Republic; MSD, Denmark; MSD, Finland; MSD, France; MSD, Ireland; MSD, Japan; MSD, Norway; MSD, Peru; MSD, Sweden; MSD Argentina, Argentina; MSD Belgium, Belgium; MSD Merck Sharp & Dohme, Germany
  • Isentress (Merck Sharp & Dohme
    China MSD, China
  • Isentress 100mg
    MSD, Switzerland
  • Isentress 25mg
    MSD, Switzerland
  • Isentress 400mg
    Merck Sharp & Dohme, Austria; Merck Sharp & Dohme, Israel; MSD, Switzerland; MSD Belgium, Luxembourg; MSD Pharma, Hungary
  • Isentress 600mg
    Merck Sharp & Dohme, Austria; MSD Belgium, Luxembourg
  • Isentress HD
    Merck Canada, Canada; Merck Sharp & Dohme, Australia

Glossary

TermDefinition
BANBritish Approved Name
BANMBritish Approved Name (Modified)
IUPACInternational Union of Pure and Applied Chemistry
ISInofficial Synonym
JANJapanese Accepted Name
OSOfficial Synonym
PHPharmacopoeia Name
Rec.INNRecommended International Nonproprietary Name (World Health Organization)
USANUnited States Adopted Name
WHOWorld Health Organization

Further information on drug naming conventions: International Nonproprietary Names.

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Further information

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