Ketoconazole Drug Interactions

ketoconazole is known to interact with the following drugs:

Click on a link below to view Drug-Drug Interactions with ketoconazole.

Major Interaction Major Interactions
Actiq, Alfenta, alfentanil, alfuzosin, alfuzosin extended release, alprazolam, alprazolam extended release, Altocor, Altoprev, amiodarone, astemizole, atorvastatin, Baycol, Camptosar, Cardioquin, cerivastatin, Cholestin (obsolete), cisapride, colchicine, conivaptan, Cordarone, Cordarone I.V., D.H.E. 45, dasatinib, dihydroergotamine, dihydroergotamine nasal, dofetilide, Duragesic, Duragesic-100, Duragesic-12, Duragesic-25, Duragesic-50, Duragesic-75, E-Mycin, E.E.S. Granules, E.E.S.-200, E.E.S.-400, E.E.S.-400 Filmtab, eletriptan, eplerenone, Ergomar, ergonovine, ergotamine, Ergotrate Maleate, Ery-Tab, Eryc, EryPed, EryPed 200, EryPed 400, Erythrocin Lactobionate, Erythrocin Stearate Filmtab, Erythrocot, erythromycin, erythromycin base, erythromycin estolate, erythromycin ethylsuccinate, erythromycin lactobionate, erythromycin stearate, fentanyl, fentanyl topical, Fentora, FK506, Halcion, Halfan, halofantrine, Hismanal, Ilosone, Ilotycin Gluceptate, Inspra, Ionsys, irinotecan, Levitra, levomethadyl acetate, Lipitor, lovastatin, lovastatin extended release, Methergine, methylergonovine, methysergide maleate, Mevacor, midazolam, Migranal, monascus, MY-E, nilotinib, Niravam, Orap, Orlaam, Pacerone, PCE Dispertab, pimozide, Prograf, Propulsid, Quin-G, Quin-Release, Quinaglute Dura-Tabs, Quinidex Extentabs, quinidine, quinidine extended release, Quinora, Ranexa, ranolazine, Rapamune, red yeast rice, Relpax, Revatio, Robimycin, salmeterol, Sansert, Serevent, Serevent Diskus, sildenafil, simvastatin, sirolimus, Sprycel, Sublimaze, tacrolimus, Tasigna, terfenadine, Tikosyn, triazolam, Uroxatral, Vaprisol, vardenafil, Versed, Viagra, Xanax, Xanax XR, Zocor

Moderate Interaction Moderate Interactions
A-Hydrocort, A-Methapred, A-Spas S/L, Abilify, Abilify Discmelt, Abraxane, Accupril, Acetocot, acetoHEXAMIDE, Acid Relief, Aciphex, Actos, Adalat, Adalat CC, Adbeon, Adgyn Estro, Adlone-40, Adlone-80, Adrenocot, Adrenocot L.A., AeroBid, AeroBid-M, Aerodiol, Afeditab CR, Agenerase, Akineton HCl, aliskiren, Alka-Mints, Alkets, Alkums, almotriptan, Aloh-Gel, Alora, alosetron, Alternagel, Alu-Cap, Alu-Tab, aluminum carbonate, aluminum hydroxide, Alvesco, Amaryl, ambrisentan, Amen, Amilac, Amitone, amitriptyline, amlodipine, Amphojel, amprenavir, Anaspaz, anisindione, aprepitant, Aptivus, Aquest, Arava, aripiprazole, Aristocort, Aristocort For Injection, Aristocort Forte, Aristopak, Aristospan Injection, Artane, atazanavir, Atreza, AtroPen, atropine, Avandia, Aventyl HCl, Avodart, Avonex, Avonex Prefilled Syringe, Axert, Axid, Axid AR, Axid Pulvules, Aygestin, Azmacort, Basaljel, beclomethasone, Beclovent, Bedol, belladonna, Belladonna Tincture, Bentyl, benztropine, bepridil, Beta-Phos/AC, betamethasone, betamethasone acet-betamethasone na phosphate, betamethasone sodium phosphate, Betaseron, bexarotene, Bextra, biperiden, bortezomib, bosentan, Bubbli-Pred, budesonide, Buprenex, buprenorphine, BuSpar, BuSpar Dividose, busPIRone, busulfan, Busulfex, Cal Oys, Cal-Gest, Calan, Calan SR, Calcarb, Calci Mix, Calci-Chew, Calcitab, calcium carbonate, Calcium Concentrate, Calcium Liquid Softgel, Calcium Oyster, Calcium Oyster Shell, Caltrate, Caltro, Camila, Cantil, carbamazepine, carbamazepine extended release, Carbatrol, Cardene, Cardene IV, Cardene SR, Cardizem, Cardizem CD, Cardizem LA, Cardizem Monovial, Cardizem SR, Cardoxin, Cartia XT, Celestone, Celestone Phosphate, Celestone Soluspan, Celexa, Cell-U-Jec, Cenestin, Cerebyx, cevimeline, chlorotrianisene, chlorproPAMIDE, Chooz, Cialis, ciclesonide, ciclesonide nasal, cilostazol, cimetidine, cinacalcet, citalopram, clidinium, Climara, Climaval, Climodien, Clinacort, Clinagen LA 40, Clinalog, clofarabine, Clolar, Cogentin, Colocort, Concentrated Phillips Milk of Magnesia, conjugated estrogens, conjugated estrogens synthetic A, conjugated estrogens synthetic B, conjugated estrogens topical, Cort-K, Cortastat, Cortastat 10, Cortastat LA, Cortef, Cortenema, Cortifoam, cortisone, Cortone Acetate, Cotolone, Coumadin, Covera-HS, Crinone, Crixivan, Curretab, Cyclogest, cycloSPORINE, Cycrin, Cystospaz, Cystospaz-M, Dalalone, Dalalone D.P., Dalalone L.A., dalfopristin, darifenacin, darunavir, ddI, De-Sone LA, Decadron, Decadron 5-12 Pak, Decadron Phosphate, Injectable, Decadron-LA, Decaject, Decaject L.A., delavirdine, Delestrogen, DELIDOSE, Delta-Lutin, Deltasone, Dep Gynogen, Dep Medalone 80, Depmedalone, Depo-Estradiol, Depo-Medrol, Depo-Predate (obsolete), Depo-Provera, Depo-Provera Contraceptive, depo-subQ provera 104, Depogen, Depoject-80, Depopred, Dermestril, Dermestril - Septem, DERMESTRIL SEPTEM, desogestrel, Desyrel, Desyrel Dividose, Detrol, Detrol LA, Dewees Carminative, Dexacen-4, Dexacort Phosphate in Respihaler, Dexacort-LA, Dexacorten, dexamethasone, dexamethasone acetate, Dexamethasone Intensol, dexamethasone sodium phosphate, Dexasone, Dexasone LA, Dexone, Dexone LA, DexPak 10 Day Taperpak, DexPak 13 DayTaperpak, Dexpak Jr. Taperpak, Di-Phen, DiaBeta, Diabinese, Dialume, Dicarbosil, dicumarol, Dicyclocot, dicyclomine, didanosine, didanosine delayed release capsule, dienestrol topical, diethylstilbestrol, Digitek, digoxin, digoxin capsule, dihydroxyaluminum sodium carbonate, Dilacor XR, Dilantin, Dilantin Infatabs, Dilantin Kapseals, Dilantin-125, Diltia XT, diltiazem, diltiazem 24 hour extended release, diltiazem extended release, Diltiazem Hydrochloride CD, Diltiazem Hydrochloride SR, Diltiazem Hydrochloride XR, Diltiazem Hydrochloride XT, Dioval 40, Dioval XX, Diskets, disopyramide, disopyramide extended release, Ditropan, Ditropan XL, Divigel 0.25 mg/packet, Divigel 0.5 mg/packet, Divigel 1 mg/packet, docetaxel, Dolophine, Donnamar, drospirenone, Dura-Estrin, Duragen, Duralone, Duralutin, dutasteride, Dymelor, Dynacirc, Dynacirc CR, echinacea, efavirenz, Elavil, Elestrin, Elleste Solo, Emend, Emend 3-Day, Emend for Injection, Enablex, Endep, Endometrin, Enjuvia, Entocort, Entocort EC, Epitol, Equetro, Equilet, erlotinib, Errin, Esclim, esomeprazole, esterified estrogens, Estinyl, Estra-C, Estra-V 40, Estrace, Estrace Vaginal Cream, Estraderm, Estraderm MX, Estraderm TTS, estradiol, estradiol acetate, estradiol benzoate, estradiol cypionate, ESTRADIOL G GAM, Estradiol Patch, estradiol topical, estradiol valerate, Estradot, Estradot 100, Estradot 37.5, Estradot 50, Estradot 75, Estragyn 5, Estragyn LA 5, ESTRAPATCH, Estrasorb, ESTREVA, Estring, Estro-A, Estro-Cyp, Estro-L.A., Estro-Span 40, Estrofem, Estrogel, estrone, Estrone AQ, estropipate, estropipate topical, eszopiclone, ethinyl estradiol, ethotoin, ethynodiol, etonogestrel, etravirine, Evamist, Evorel, Evoxac, Ex-Lax Milk of Magnesia, Extra Strength Mylanta Calci Tabs, famotidine, Fareston, felodipine, felodipine extended release, Fematrix, Fempatch, Femring, FEMSEPT, FemSeven, FemSeven Sequi Phase I, FemTab, Femtrace, Femtran, First Progesterone MC10, First Progesterone MC5, FIRST-Progesterone VGS 100, FIRST-Progesterone VGS 200, FIRST-Progesterone VGS 25, FIRST-Progesterone VGS 400, FIRST-Progesterone VGS 50, flavoxate, Flo-Pred, Flonase, Florinef Acetate, Flovent, Flovent Diskus, Flovent HFA, Flovent Rotadisk, fludrocortisone, flunisolide, fluticasone, fluticasone nasal, fluvoxamine, fluvoxamine extended release, Folex PFS, Fortovase, fosamprenavir, fosaprepitant, fosphenytoin, Fosrenol, galantamine, galantamine extended release, gefitinib, Gengraf, Gestone, Gleevec, glimepiride, glipiZIDE, glipiZIDE extended release, GlipiZIDE XL, Glucotrol, Glucotrol XL, glyBURIDE, glyBURIDE micronized, glycopyrrolate, Glynase PresTab, grepafloxacin, Gynodiol, Gynogen LA 20, Heartburn Relief, Hexadrol, Hexadrol Phosphate, homatropine, Hydeltra-T.B.A., Hydeltrasol, hydrocortisone, hydrocortisone acetate, hydrocortisone cypionate, hydrocortisone hemisuccinate, hydrocortisone sodium phosphate, Hydrocortisone Sodium Succinate, Hydrocortone, Hydrocortone Phosphate, hydroxyprogesterone, Hylutin, HyoMax DT, HyoMax FT, HyoMax SL, HyoMax SR, hyoscyamine, hyoscyamine extended release, Hyosol, Hyospaz, Hyosyne, Hyprogesterone, IB-Stat, Icar Prenatal Chewable Calcium, imatinib, imipramine, imipramine pamoate, Implanon, indinavir, INH, Intelence, interferon beta-1a, interferon beta-1b, Invirase, Iressa, isoniazid, Isoptin, Isoptin I.V., Isoptin SR, isradipine, isradipine extended release, ixabepilone, Ixempra, Jantoven, Jolivette, Kemadrin, Ken-Jec 40, Kenaject-40, Kenalog-10, Kenalog-40, Kestrone 5, Key-Pred, Key-Pred SP, L-hyoscyamine, Lanoxicaps, Lanoxin, lansoprazole, lanthanum carbonate, lapatinib, Lariam, Leader Acid Reducer, leflunomide, Letairis, Levbid, levonorgestrel, Levsin, Levsin SL, Levsinex SR, Lexiva, Liquid Pred, Losospan, Lotronex, Lowsium, Luminal, Lunesta, Luvox, Luvox CR, M-PREDNISolone, Maalox Antacid Barrier, Maalox Childrens', Maalox Quick Dissolve, Maalox Quick Dissolve Extra Strength, Maalox Quick Dissolve Maximum Strength, Maalox Regular Strength, Mag-200, Mag-Carb, Mag-Ox 400, magaldrate, MagGel, magnesium carbonate, magnesium hydroxide, magnesium oxide, magnesium trisilicate, Maldemar, Maoson, maraviroc, Med-Jec-40, Medicort, Medidex, Medidex LA, Medidiol 10, Medipred, Medralone, Medralone 40, Medralone 80, Medrol, Medrol Dosepak, medroxyPROGESTERone, mefloquine, Menaval-20, Menest, Menopause Formula Progesterone, MENOREST, Menorest Patch, Menostar, mepenzolate, mephenytoin, Mesantoin, mestranol, Methacort 40, Methacort 80, methadone, Methadose, methotrexate, Methotrexate Sodium, Preservative Free, methscopolamine, Methylcotol, Methylcotolone, Methylpred DP, methylPREDNISolone, methylPREDNISolone acetate, MethylPREDNISolone Dose Pack, methylPREDNISolone sodium succinate, Meticorten, Mg hydroxide, Mg oxide, mibefradil, Micronase, Milk of Magnesia, Millipred, Miradon, Mirena, Mycobutin, Mylanta AR, Mylanta Child, Myleran, naltrexone, nefazodone, Neoral, Nephro Calci, Neut, nevirapine, Nexium, Nexium I.V., niCARdipine, niCARdipine extended release, Nifediac CC, Nifedical XL, NIFEdipine, NIFEdipine extended release, nimodipine, Nimotop, nisoldipine, nizatidine, Nor-QD, Nora-Be, norelgestromin, norethindrone, norethindrone acetate, norethindrone topical, norgestimate, norgestrel, Norpace, Norpace CR, Norplant System, nortriptyline, Norvasc, Norvir, Norvir Soft Gelatin, Nulev, Nuvelle TS Phase I, Nydrazid, Oesclim, Oestradiol, Oestradiol Implants, OESTRODOSE, OESTROGEL, Oestrogel Pump-Pack, Ogen 0.625, Ogen 1.25, Ogen 2.5, Ogen Vaginal Cream, omeprazole, Omnaris, Onxol, Orapred, Orapred ODT, Orasone, Organon Oestradiol, Orinase, Orion Progesterone, OROMONE, Ortho Dienestrol, Ortho Micronor, Ortho-Est, Os-Cal, Os-Cal 500, Ovrette, oxcarbazepine, oxybutynin, oxybutynin extended release, Oxytrol, Oysco 500, Oyst Cal, Oyst Cal 500, Oyster, Oyster Cal, Oyster Cal 500, Oyster Calcium, Oyster Shell, oyster shell calcium, Oyster Shell Calcium 500, paclitaxel, paclitaxel protein-bound, Pamelor, Pamine, Pamine Forte, pantoprazole, paricalcitol, Pediapred, Peganone, Pepcid, Pepcid AC, Pepcid AC Maximum Strength, Pepcid RPD, Pepto Children's, phenobarbital, Phenytek, phenytoin, phenytoin extended release, Phenytoin Sodium, Prompt, Phillips Milk of Magnesia, Phillips' Cramp-free, pioglitazone, Plan B, Plendil, Pletal, Posicor, Prandin, Pred-Ject-50, Predacort 50, Predacorten, Predaject-50, Predalone 50, Predate-50, Predcor, Predicort RP, Predicort-50, Prednicen-M, Prednicot, prednisoLONE, prednisoLONE acetate, prednisoLONE sodium phosphate, prednisoLONE tebutate, predniSONE, Prelone, Premarin, Premarin Intravenous, Premarin Vaginal, Prevacid, Prevacid I.V., Prevacid SoluTab, Prezista, Pri-Cortin 50, Priftin, Prilosec, Prilosec OTC, Primethasone, Primogyn Depot, Pro-Banthine, Procardia, Procardia XL, Prochieve, procyclidine, Prodrox, Progest, Progestasert System, progesterone, progesterone topical, Progynova, Progynova TS, Prometrium, propantheline, Protonix, Protonix IV, PROVAMES, Provera, Pulmicort Flexhaler, Pulmicort Nebuamp, Pulmicort Respules, Pulmicort Turbuhaler, Quarzan, quetiapine, quetiapine extended release, quinapril, quinestrol, Qvar, rabeprazole, ramelteon, ranitidine, ranitidine bismuth citrate, Raxar, Razadyne, Razadyne ER, Rebif, Regurin, Reminyl, repaglinide, Rescriptor, ReVia, Reyataz, Rezulin, Rheumatrex Dose Pack, Ri-Mag, rifabutin, Rifadin, Rifadin IV, rifampin, rifapentine, Rimactane, Riopan, ritonavir, Robinul, Robinul Forte, Rolaids Sodium Free, Rolaids Soft Chew, Ron Acid, rosiglitazone, Rozerem, Sal-Tropine, Sanctura, Sanctura XR, Sandimmune, Sandrena, saquinavir, saquinavir mesylate, Scopace, scopolamine, scopolamine topical, Selestoject, Selzentry, Sensipar, Seroquel, Seroquel XR, Serzone, sodium bicarbonate, Solfoton, solifenacin, Solu-Cortef, Solu-Medrol, Solurex, Solurex LA, Spasdel, Sterapred, Sterapred DS, Stilphostrol, Subutex, Sufenta, sufentanil, Sular, sunitinib, Super Calcium, Surpass, Surpass Extra Strength, Sustiva, Sutent, Symax Duotab, Symax FasTab, Symax SL, Symax SR, SYSTEN, TAC 3, Tace, tadalafil, Tagamet, Tagamet HB, Tarceva, Targretin, Taxol, Taxotere, Taztia XT, Tegretol, Tegretol XR, Tekturna, Telzir, temsirolimus, THAIS, THAISSEPT, thioguanine, Tiazac, tipranavir, Titralac, Tofranil, Tofranil-PM, Tol-Tab, TOLAZamide, TOLBUTamide, Tolinase, tolterodine, tolterodine extended release, toremifene, Torisel, Tracleer, Tramacort-D, Transderm-Scop, traZODONE, Trexall, Triam-A, Triam-Forte, triamcinolone, triamcinolone acetonide, triamcinolone diacetate, triamcinolone hexacetonide, triamcinolone ophthalmic, Triamcot, Triamonide 40, Triesence, Trihexane, trihexyphenidyl, Trileptal, Trilog, Trilone, Tristoject, Tritec, troglitazone, trospium, trospium extended release, Tums, Tums 500, Tums E-X, Tums Extra Strength, Tums Ultra, Tykerb, U-Tri-Lone, Ultra Mylanta Calci Tabs, Urispas, Uro-Mag, Urotrol, Vagifem, valdecoxib, Valergen, Vanatrip, Vanceril, Vanceril DS, Vascor, Velcade, Veramyst, verapamil, verapamil 24 hour extended release, verapamil extended release, Verelan, Verelan PM, VESIcare, VFEND, Videx, Videx EC, Viramune, Vivelle, Vivelle-Dot, VIVELLEDOT, Vivitrol, voriconazole, warfarin, Zantac, Zantac 150, Zantac 300, Zantac 300 GELdose, Zantac 75, Zantac EFFERdose, Zantac GELdose, Zegerid (Original Formulation), Zemplar, Zonegran, zonisamide, Zumenon

Minor Interaction Minor Interactions
Abelcet, Aerius, Aerolate III, Aerolate JR, Aerolate SR, Alavert, alcohol, alcohol, ethyl, Allegra, Allegra ODT, Altabax, Ambien, Ambien CR, AmBisome, aminophylline, aminophylline extended release, Amphocin, Amphotec, amphotericin B, amphotericin B cholesteryl sulfate, amphotericin B lipid complex, amphotericin B liposomal, Aquaphyllin, Aricept, Aricept ODT, armodafinil, Asmalix, Asmanex Twisthaler 120 Dose, Asmanex Twisthaler 14 Dose, Asmanex Twisthaler 30 Dose, Asmanex Twisthaler 60 Dose, Basic Vitamins Brewers Yeast, brewer's yeast, Bronkodyl, Carafate, Choledyl, Choledyl SA, Clarinex, Clarinex Reditabs, Claritin, Claritin 24 Hour Allergy, Claritin Hives Relief, Claritin Reditab, Clear-Atadine, Clear-Atadine Children's, Cozaar, Dehydrated Alcohol, desloratadine, Dimetapp ND, donepezil, Elidel, Elixophyllin, ethanol, Ethyl Alcohol, fexofenadine, Fungizone, Fungizone For Tissue Culture, Geodon, granisetron, Granisol, Ketek, Ketek Pak, Kytril, lopinavir, loratadine, Loratadine Reditab, losartan, Major Brewers Yeast, Marlex Brewers Yeast, Mason Vitamins Brewers Yeast, Meridia, Mifeprex, mifepristone, modafinil, mometasone, montelukast, Naropin, Naropin Novaplus, Naropin Polyamp, Naropin SDV, Natures Bounty Brewers Yeast, Natures Naturals Brewers Yeast, nelfinavir, Neoclarityn, NeuTrexin, Nuvigil, Oncovin, oxtriphylline, oxtriphylline extended release, pimecrolimus topical, Provigil, Quibron-T, Quibron-T/SR, Respbid, retapamulin topical, ropivacaine, RU-486, sibutramine, Singulair, Slo-Bid Gyrocaps, Slo-Phyllin, Slo-Phyllin 125, Slo-Phyllin 80, sucralfate, T-Phyl, Tavist ND, telithromycin, Theo-24, Theo-Dur, Theo-Dur Sprinkles, Theo-Time, Theo-X, Theobid, TheoCap, Theochron, Theoclear L.A.-130, Theoclear L.A.-260, Theoclear-80, Theolair, Theolair-SR, theophylline, theophylline 24 hr extended release, theophylline extended release, Theovent, trimetrexate, Truphylline, Truxophyllin, Uni-Dur, Uniphyl, Velban, vinBLAStine, Vincasar PFS, vinCRIStine, Viracept, Wal-itin, ziprasidone, zolpidem, zolpidem extended release

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